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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T41319 D-Saccharic acid 1,4-lactone hydrate

Others Others
D-Saccharic acid 1,4-lactone hydrate 是β-葡萄糖醛酸酶的有效抑制剂(IC50=48.4 μM),可用作标准药物。D-Saccharic acid 1,4-lactone hydrate 显示出抗癌、解毒和抗氧化的活性性。
T35454 γ-Glu-Cys (ammonium salt)

γ-Glu-Cys is an intermediate in glutathione (GSH) synthesis.1It is formed by ATP-dependent condensation of cysteine and glutamate by γ-glutamylcysteine synthetase. γ-Glu-Cys is also an essential component of phytochelatins, the heavy metal detoxifying enzymes in plants.2
T78032 Endotoxin inhibitor TFA

Endotoxin inhibitor TFA 是一种可以与脂多糖(LPS)的成分脂质A高亲和力结合的合成肽,具有中和LPS毒性、预防LPS引发的细胞因子释放的作用。此外,Endotoxin inhibitor TFA能够有效抑制LPS引起的发热反应,同时具有极低的毒性和致死率。

化合物

D-Saccharic acid 1,4-lactone hydrate
Cat.No: T41319
Synonym:
Target: Others
γ-Glu-Cys (ammonium salt)
Cat.No: T35454
Synonym:
Target:
Endotoxin inhibitor TFA
Cat.No: T78032
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T0928 L-Ascorbic acid

维生素C,Vitamin C,Ascorbic acid,L(+)-Ascorbic acid,抗坏血酸,L-Ascorbate

Apoptosis; Calcium Channel; Reactive Oxygen Species; Endogenous Metabolite Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB
L-Ascorbic acid (Vitamin C) 属于天然产物,是一种强效的还原剂和抗氧化剂。L-Ascorbic acid 具有抗细菌感染、解毒反应和胶原蛋白形成的作用。L-Ascorbic acid 被用于治疗坏血病。
TJO2758 D-Glucuronic acid

D-葡萄糖醛酸,Aldehydo-D-Glucuronic Acid

Others; Endogenous Metabolite Metabolism; Others
D-Glucuronic acid (Aldehydo-D-Glucuronic Acid) 是一种从许多树胶中分离出的重要中间体。它对皮肤具有抗炎作用。它及其衍生物葡萄糖醛酸内酯作为预防人类健康的肝脏解毒剂。

天然产物

L-Ascorbic acid
Cat.No: T0928
Synonym: 维生素C,Vitamin C,Ascorbic acid,L(+)-Ascorbic acid,抗坏血酸,L-Ascorbate
Target: Apoptosis, Calcium Channel, Reactive Oxygen Species, Endogenous Metabolite
D-Glucuronic acid
Cat.No: TJO2758
Synonym: D-葡萄糖醛酸,Aldehydo-D-Glucuronic Acid
Target: Others, Endogenous Metabolite
TargetMol Loading
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