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Cat. No. Product Name Target Signaling Pathways
T2583 Cilastatin

西司他丁,MK0791

Proteasome; Antibacterial; Antibiotic Microbiology/Virology; Proteases/Proteasome; Ubiquitination
Cilastatin (MK0791) 是一种可逆的竞争性的肾脏脱氢肽酶 I 抑制剂,IC50为 0.1 μM。它抑制细菌金属叶内酰胺酶CphA 的IC50为 178 μM,可用作抗菌辅助剂。
T6411 Biapenem

CLI 86815,比阿培南,Biapenern,Omegacin,L 627,LJC 10627

Antibacterial; Antibiotic Microbiology/Virology
Biapenem (CLI 86815) 是不经肠道的广谱碳青霉烯抗生素。
T2583L Cilastatin sodium

Cilastatinum,Cilastatin Monosodium Salt ;Cilastatin Sodium,Cilastatin Monosodium Salt,MK 791,Cilastatine,Cilastatin,Cilastatin Sodium,MK 0791

Cilastatin is a renal dehydropeptidase-I and leukotriene D4 dipeptidase inhibitor.
T33441 MK789

MK 789,MK-789

MK-789 is an inhibitor of dehydropeptidase I. MK-789 and MK-791 alter the renal excretion of N-formimidoyl thienamycin from glomerular filtration plus tubular secretion to glomerular filtration only, possibly by competitively inhibiting the penetration of
T71317 WS1358A1 disodium

WS1358A1 disodium is a potent inhibitor of renal dehydropeptidase.
T23939 DA 1131

DA-1131,DA1131

DA 1131 is a new carbapenem antibiotic. It undergoes renal metabolism by renal dehydropeptidase I.

化合物

Cilastatin
Cat.No: T2583
Synonym: 西司他丁,MK0791
Target: Proteasome, Antibacterial, Antibiotic
Biapenem
Cat.No: T6411
Synonym: CLI 86815,比阿培南,Biapenern,Omegacin,L 627,LJC 10627
Target: Antibacterial, Antibiotic
Cilastatin sodium
Cat.No: T2583L
Synonym: Cilastatinum,Cilastatin Monosodium Salt ;Cilastatin Sodium,Cilastatin Monosodium Salt,MK 791,Cilastatine,Cilastatin,Cilastatin Sodium,MK 0791
Target:
MK789
Cat.No: T33441
Synonym: MK 789,MK-789
Target:
WS1358A1 disodium
Cat.No: T71317
Synonym:
Target:
DA 1131
Cat.No: T23939
Synonym: DA-1131,DA1131
Target:
TargetMol Loading
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