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Cat. No. Product Name Target Signaling Pathways
T9066 Merafloxacin

CI 934

SARS-CoV Microbiology/Virology
Merafloxacin (CI 934) 是一种氟喹诺酮类抗菌药物,也被确定为 SARS-CoV-2 的 1 PRF 抑制剂。它对革兰氏阳性菌和革兰氏阴性菌具有体外活性。
T8688 (Rac)-X77

CPD77,MUN91789

SARS-CoV Microbiology/Virology
(Rac)-X77 (MUN91789) 是一种 SARS-​CoV-​2 主要蛋白酶抑制剂。
T8309 EIDD-2801

Molnupiravir

SARS-CoV Microbiology/Virology
EIDD-2801 (Molnupiravir) 是核糖核苷类似物 N 4-羟基胞苷 (EIDD-1931) 的异丙酯前药,已显示出广泛的流感病毒和多种冠状病毒活性。
T18911 Acriflavine

Acriflavinium chloride 3,6-Acridinediamine mix

SARS-CoV; Antibacterial Microbiology/Virology
Acriflavine (Acriflavinium chloride 3,6-Acridinediamine mix) 是木瓜蛋白酶样蛋白酶(PL(pro))抑制剂,是一种用于标记高分子量 RNA 的荧光染料,具有抗菌抗癌活性,抑制 SARS-CoV-2 和其他 β 冠状病毒,可用于研究白血病。
T60951 Molnupiravir

EIDD-2801,Lagevrio,MK-4482

SARS-CoV; Influenza Virus Microbiology/Virology
Molnupiravir (MK-4482) (EIDD-2801) 是核糖核苷类似物 EIDD-1931 的异丙酯前体药物,具有口服生物利用度。Molnupiravir 可用于 COVID-19 ,季节性和流行性流感的研究,对多种冠状病毒和流感病毒具有广谱的抗病毒活性,例如,SARS-CoV-2,MERS-CoV,SARS-CoV。
T69868 ZIKV-IN-K22

ZIKV-IN-K22 is a potent antiviral agent against a broad range of coronaviruses by targeting membrane-bound viral RNA replication, effectively inhibiting ZIKV with IC50 of 2.1 μM.
T82948 Atilotrelvir

Atilotrelvir 为一种抗病毒药物,能够抑制冠状病毒、小核糖核酸病毒及诺如病毒的感染。
T41177 Galidesivir dihydrochloride

BCX 4430

Galidesivir is a viral RNA-dependent RNA polymerase (RdRP) inhibitor and broad spectrum antiviral nucleotide.In vitro, galidesivir displays antiviral activity against a range of RNA viruses, including bunyaviruses, arenaviruses, paramyxoviruses, coronaviruses, and flaviviruses (EC50values range from 3 μM to >100 μM). Galidesivir protects against Ebola and Marburg viral infection in animal models.
T76900 Adintrevimab

Adintrevimab (ADG 20),一种人IgG1单克隆抗体,针对SARS-CoV(SARS-CoV)。它能抑制SARS-CoV-2变体及其他具有大流行潜力的SARS样冠状病毒。
T63537 SARS-CoV-2 3CLpro-IN-1

SARS-CoV-2 3CLpro-IN-1 (Compound 14c) is a highly potent inhibitor specifically designed to target and inhibit the activity of SARS-CoV-2 3CL pro, which is a cysteine-protease found in the main coronaviruses. This particular enzyme has been recognized as a highly promising target for the development of effective antiviral drugs. Therefore, SARS-CoV-2 3CLpro-IN-1 holds significant potential for advancing research and development in the field of infectious diseases [1].
T78867 WU-04

SARS-CoV Microbiology/Virology
WU-04为针对SARS-CoV-2的3CLpro蛋白的非共价抑制剂,对包括Alpha、Beta、Gamma、Delta、Lambda和Omicron在内的6种SARS-CoV-2变体及SARS-CoV与MERS-CoV的3CLpro蛋白展现出高效的抑制作用。
T72312 SARS-CoV-2 3CLpro-IN-10

SARS-CoV-2 3CLpro-IN-10(5d)为一种有效的抗 SARS-CoV-2 3CL 蛋白酶抑制剂,其IC50值仅为190 nM,同时对SARS-CoV-1的IC50值为790 nM,对MERS-CoV的IC50值则为70 nM,显示出广谱的抗病毒活性。
T38174 Mpro inhibitor N3 hemihydrate

Mpro inhibitor N3 hemihydrate is a potent inhibitor of SARS-CoV-2 Mpro with an EC50 of 16.77 μM for SARS-CoV-2. Mpro inhibitor N3 hemihydrate specifically inhibits Mpro from multiple coronaviruses, including SARS-CoV and MERS-CoV. Mpro inhibitor N3 hemihydrate displays inhibition against HCoV-229E, FIPV, and MHV-A59 with individual IC50 of 4.0 μM, 8.8 μM, and 2.7 μM, respectively[1][2]. Mpro inhibitor N3 hemihydrate (0-0.64 μM) is able to penetrate cells to inhibit the replication of IBV viruses...

化合物

Merafloxacin
Cat.No: T9066
Synonym: CI 934
Target: SARS-CoV
(Rac)-X77
Cat.No: T8688
Synonym: CPD77,MUN91789
Target: SARS-CoV
EIDD-2801
Cat.No: T8309
Synonym: Molnupiravir
Target: SARS-CoV
Acriflavine
Cat.No: T18911
Synonym: Acriflavinium chloride 3,6-Acridinediamine mix
Target: SARS-CoV, Antibacterial
Molnupiravir
Cat.No: T60951
Synonym: EIDD-2801,Lagevrio,MK-4482
Target: SARS-CoV, Influenza Virus
ZIKV-IN-K22
Cat.No: T69868
Synonym:
Target:
Atilotrelvir
Cat.No: T82948
Synonym:
Target:
Galidesivir dihydrochloride
Cat.No: T41177
Synonym: BCX 4430
Target:
Adintrevimab
Cat.No: T76900
Synonym:
Target:
SARS-CoV-2 3CLpro-IN-1
Cat.No: T63537
Synonym:
Target:
WU-04
Cat.No: T78867
Synonym:
Target: SARS-CoV
SARS-CoV-2 3CLpro-IN-10
Cat.No: T72312
Synonym:
Target:
Mpro inhibitor N3 hemihydrate
Cat.No: T38174
Synonym:
Target:
TargetMol Loading
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