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Cat. No. Product Name Target Signaling Pathways
T4170 PKM2-IN-1

PKM2 inhibitor,compound 3k

PKM Metabolism
PKM2-IN-1 (compound 3k) 是丙酮酸激酶 M2 (PKM2) 抑制剂,其IC50=2.95 μM。
T61226 hDHODH-IN-9

hDHODH-IN-9 (Compound 3k) is a highly potent inhibitor of hDHODH, exhibiting an IC50 of 0.34 μM. It displays significant cytotoxic activity against MCF-7 and A375 cells, while maintaining good selectivity. With its characteristics, hDHODH-IN-9 holds promise for cancer disease research [1].
T60465 Anti-infective agent 2

Anti-infective agent 2 (化合物 3k) 是一种抗原生动物和抗分枝杆菌剂。Anti-infective agent 2对P. falciparum 和T. brucei rhodesiense 显示出抗寄生虫活性,IC50值分别为 0.07 和 2.20 μM。Anti-infective agent 2 对耻垢分枝杆菌显示出抗分支杆菌活性,其MIC 为 32 μg/mL。

化合物

PKM2-IN-1
Cat.No: T4170
Synonym: PKM2 inhibitor,compound 3k
Target: PKM
hDHODH-IN-9
Cat.No: T61226
Synonym:
Target:
Anti-infective agent 2
Cat.No: T60465
Synonym:
Target:
TargetMol Loading
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