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3

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T5413 ML216

CID-49852229

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
ML216 (CID-49852229) 是一种选择性、细胞渗透性的BLM 解旋酶抑制剂,具有抗肿瘤活性。它对BLMfull-length 和BLM636-1298的IC50分别为 2.98 μM 和 0.97 μM。
T68428 ZK-Thiazolidinone

ZK-Thiazolidinone, also known as TAL, is an ATP-competitive inhibitor of PLK1. In vitro, ZK-Thiazolidinone counteracts the role of Plk1 in previously established functions, notably, sister chromatid separation, centrosome maturation, and bipolar spindle assembly. In vivo, ZK-Thiazolidinone selectively inhibits PLK1 and causes a prometaphase-like mitotic (G2–M) arrest. ZK-Thiazolidinone inhibits human PLK1 (IC50, 19± 12 nM) and various human and mouse tumor cell lines (IC50, 0.2–1.3 μM). ZK-Thiaz...
T83829 2'-Deoxy-1,N6-ethenoadenosine-5'-O-triphosphate sodium

ε-dATP

ε-dATP是一种具有荧光性的嘌呤核苷酸2’-脱氧腺苷-5’-O-三磷酸(dATP)衍生物。它能在50至150µM的浓度范围内诱导初级小鼠脾脏T细胞和B细胞在脂多糖(LPS)或刀豆蛋白A刺激下发生姊妹染色单体交换。ε-dATP已被用于研究乙烯氯诱导的突变过程中模糊碱基配对的情况。相关的ATP衍生物ε-ATP,在300 nm激发下显示415 nm的发射峰值。

化合物

ML216
Cat.No: T5413
Synonym: CID-49852229
Target: DNA/RNA Synthesis
ZK-Thiazolidinone
Cat.No: T68428
Synonym:
Target:
2'-Deoxy-1,N6-ethenoadenosine-5'-O-triphosphate sodium
Cat.No: T83829
Synonym: ε-dATP
Target:
Cat. No. Product Name Target Signaling Pathways
T4730 Thymidine-5'-monophosphate disodium salt

胸苷酸二钠,Thymidine 5'-monophosphate disodium salt,TMP DISODIUM SALT

Others; Endogenous Metabolite Metabolism; Others
Thymidine-5'-monophosphate disodium salt (TMP DISODIUM SALT) 是内源性代谢产物的一种。
TN1138 γ-Fagarine

γ-崖椒碱,gamma-Fagarine

HCV Protease Microbiology/Virology; Proteases/Proteasome
gamma-Fagarine possesses moderate levels of anti-HCV activities with IC50 values being 20.4 ± 0.4 ug/ml, respectively. It has sister chromatid exchanges (SCEs)-inducing activity

天然产物

Thymidine-5'-monophosphate disodium salt
Cat.No: T4730
Synonym: 胸苷酸二钠,Thymidine 5'-monophosphate disodium salt,TMP DISODIUM SALT
Target: Others, Endogenous Metabolite
γ-Fagarine
Cat.No: TN1138
Synonym: γ-崖椒碱,gamma-Fagarine
Target: HCV Protease
TargetMol Loading
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