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Cat. No. | Product Name | Target | Signaling Pathways |
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T5413 |
ML216
CID-49852229 |
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
ML216 (CID-49852229) 是一种选择性、细胞渗透性的BLM 解旋酶抑制剂,具有抗肿瘤活性。它对BLMfull-length 和BLM636-1298的IC50分别为 2.98 μM 和 0.97 μM。 | |||
T68428 |
ZK-Thiazolidinone
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ZK-Thiazolidinone, also known as TAL, is an ATP-competitive inhibitor of PLK1. In vitro, ZK-Thiazolidinone counteracts the role of Plk1 in previously established functions, notably, sister chromatid separation, centrosome maturation, and bipolar spindle assembly. In vivo, ZK-Thiazolidinone selectively inhibits PLK1 and causes a prometaphase-like mitotic (G2–M) arrest. ZK-Thiazolidinone inhibits human PLK1 (IC50, 19± 12 nM) and various human and mouse tumor cell lines (IC50, 0.2–1.3 μM). ZK-Thiaz... | |||
T83829 |
2'-Deoxy-1,N6-ethenoadenosine-5'-O-triphosphate sodium
ε-dATP |
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ε-dATP是一种具有荧光性的嘌呤核苷酸2’-脱氧腺苷-5’-O-三磷酸(dATP)衍生物。它能在50至150µM的浓度范围内诱导初级小鼠脾脏T细胞和B细胞在脂多糖(LPS)或刀豆蛋白A刺激下发生姊妹染色单体交换。ε-dATP已被用于研究乙烯氯诱导的突变过程中模糊碱基配对的情况。相关的ATP衍生物ε-ATP,在300 nm激发下显示415 nm的发射峰值。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T4730 |
Thymidine-5'-monophosphate disodium salt
胸苷酸二钠,Thymidine 5'-monophosphate disodium salt,TMP DISODIUM SALT |
Others; Endogenous Metabolite | Metabolism; Others |
Thymidine-5'-monophosphate disodium salt (TMP DISODIUM SALT) 是内源性代谢产物的一种。 | |||
TN1138 |
γ-Fagarine
γ-崖椒碱,gamma-Fagarine |
HCV Protease | Microbiology/Virology; Proteases/Proteasome |
gamma-Fagarine possesses moderate levels of anti-HCV activities with IC50 values being 20.4 ± 0.4 ug/ml, respectively. It has sister chromatid exchanges (SCEs)-inducing activity |