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Cat. No. Product Name Target Signaling Pathways
T6452 Closantel Sodium

Antibacterial; Parasite Microbiology/Virology
Closantel sodium 是抗寄生虫活性的卤化水杨酰苯胺。它是高度特异性的盘尾丝虫几丁质酶抑制剂。
T0237 Closantel

氯氰碘柳胺,R-31520,氯生太尔

Antibacterial; Parasite Microbiology/Virology
Closantel (R-31520) 是抗寄生虫活性的卤化水杨酰苯胺。它是高度特异性盘尾丝虫几丁质酶抑制剂。
T40863 Bisdionin C

Antibacterial Microbiology/Virology
Bisdionin C 是一种有效的 GH18 chitinase 抑制剂,对 A. fumigatus ChiB1 的 IC50 为 0.2 μM。 Bisdionin C 抑制人巨噬细胞壳三糖苷酶 (HCHT, IC50 = 8.3 μM) 和酸性哺乳动物几丁质酶 (AMCase, IC50 = 3.4 μM)。
T9592 OATD-01

Others Others
OATD-01 是一种壳三糖苷酶及酸性哺乳动物几丁质酶的高活性抑制剂,对CHIT1具有低纳摩尔活性 (hCHIT1,IC50=23 nM)。它在多个物种中显示出良好的药代动力学特征,在体内具有显著的抗纤维化活性,可用于研究肺纤维化。
TP2140 Argifin

Others Others
Argifin is a sub-nanomolar chitinase inhibitor produced by soil microorganisms (IC50: 0.025 μM, 6.4 μM, 1.1 μM and 4.5 μM for SmChiA (Serratia marcescens chitinaese A), SmChiB, Aspergillus fumigatus chitinase B1 and human chitotriosidase).
T9952 OAT-2068

Others Others
OAT-2068 是一种有效且选择性的小鼠壳三糖苷酶 (CHIT1) 抑制剂,与 mAMCase 相比,mCHIT1 的选择性高出 143 倍。
T37570 4-Methylumbelliferyl-β-D-N,N',N''-Triacetylchitotrioside

4-Methylumbelliferyl-β-D-N,N',N''-triacetylchitotrioside is a fluorogenic substrate for chitinases and chitotriosidases. 4-Methylumbelliferyl-β-D-N,N',N''-triacetylchitotrioside is cleaved by chitinases and chitotriosidases to release the fluorescent moiety 4-methylumbelliferyl (4-MU). 4-MU fluorescence is pH-dependent with excitation maxima of 320 and 360 nm at low (1.97-6.72) and high (7.12-10.3) pH, respectively, and an emission maximum ranging from 445 to 455 nM, increasing as pH decreases. ...

化合物

Closantel Sodium
Cat.No: T6452
Synonym:
Target: Antibacterial, Parasite
Closantel
Cat.No: T0237
Synonym: 氯氰碘柳胺,R-31520,氯生太尔
Target: Antibacterial, Parasite
Bisdionin C
Cat.No: T40863
Synonym:
Target: Antibacterial
OATD-01
Cat.No: T9592
Synonym:
Target: Others
Argifin
Cat.No: TP2140
Synonym:
Target: Others
OAT-2068
Cat.No: T9952
Synonym:
Target: Others
4-Methylumbelliferyl-β-D-N,N',N''-Triacetylchitotrioside
Cat.No: T37570
Synonym:
Target:
TargetMol Loading
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