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Cat. No. | Product Name | Target | Signaling Pathways |
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T60028 | MM41 | DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
MM41 是一种人类端粒和基因启动子 DNA 四链体稳定剂,对 MIA PaCa-2 胰腺癌细胞系的 IC50 <10 nM。 | |||
T21648 |
CP-31398 dihydrochloride
CP 31398 dihydrochloride |
p53 | Apoptosis |
CP-31398 dihydrochloride 是一种 p53 稳定剂,可稳定 p53 的活性构象并促进具有突变型或野生型 p53 的癌细胞系中的 p53 活性。 | |||
T31364 |
Dehydelone
KOS1584,SK-10088,KOS-1584,R-1645,SK10088,R1645 |
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Dehydelone(KOS-1584, R-1645, SK-10088) is a microtubule stabilizer that may be used in the treatment of non-small cell lung cancer. | |||
T32419 |
KRAS4b-PDEδ stabilizer C19
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KRAS4b-PDEδ stabilizer C19 is a stabilizer of the KRAS4b-PDEδ complex which decreases the proliferation of colorectal cancer cells, and increases apoptosis via decreased activation of oncogenic KRAS4b signaling. | |||
T61024 | PK9327 | ||
PK9327 是可靶向空腔的 p53癌症突变的小分子稳定剂,。 | |||
T81285 | RGB-1 | ||
RGB-1为多环芳烃类化合物,作为RNA G-四链体 (RNA G-quadruplexes) 的稳定剂,能够抑制RNA翻译,并在乳腺癌细胞中下调NRAS原癌基因的表达。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T75573 | Taccalonolide E | ||
Taccalonolide E 是一种微管稳定剂,诱导癌细胞凋亡 (apoptosis)。 |