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3

抑制剂 & 化合物

6

天然产物

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Cat. No. Product Name Target Signaling Pathways
T37413 Calcitonin (salmon) (trifluoroacetate salt)

Calcitonin is a peptide hormone that lowers blood calcium level and inhibits bone resorption. It belongs to the calcitonin family of peptides, which also includes amylin , calcitonin gene-related peptide , and adrenomedullin. The binding of salmon calcitonin to the human calcitonin receptor (CTR) is not modulated by receptor activity-modifying proteins (RAMPs), which influence affinity of human calcitonin to CTR. Salmon calcitonin binds to human CTR2 with IC50 values of 0.933, 0.224, 0.134, and ...
TP1040 Calcitonin (salmon)

鲑降钙素,Calcitonin salmon,Salmon calcitonin

CGRP Receptor GPCR/G Protein; Neuroscience
Calcitonin (salmon) 是一种阿米林和卡西宁受体的双激动剂,是一种钙调节激素,能够刺激骨的生成并能抑制骨吸收。
TP1040L Calcitonin(salmon) Acetate(47931-85-1(free base))

Salmon calcitonin

CGRP Receptor GPCR/G Protein; Neuroscience
Calcitonin(salmon)Acetate (47931-85-1(free base))(Salmon calcitonin) 是一种钙调节激素,用于治疗绝经后至少 5 年的女性骨质疏松症。

化合物

Calcitonin (salmon) (trifluoroacetate salt)
Cat.No: T37413
Synonym:
Target:
Calcitonin (salmon)
Cat.No: TP1040
Synonym: 鲑降钙素,Calcitonin salmon,Salmon calcitonin
Target: CGRP Receptor
Calcitonin(salmon) Acetate(47931-85-1(free base))
Cat.No: TP1040L
Synonym: Salmon calcitonin
Target: CGRP Receptor
Cat. No. Product Name Target Signaling Pathways
Fr13883 3-Methoxyphenylacetic acid

Others Others
3-Methoxyphenylacetic acid 是 m-hydroxyphenylacetic (m-OHPAA) 的衍生物,茄形假丝酵母中的一种植物毒素。它可用于针对介氧菌根腐烂的毒素介导的生物测定法的开发。
T41372 (22S,23S)-Homobrassinolide

油菜素内酯,SSHB

Others Others
(22S,23S)-Homobrassinolide (SSHB) 在各种植物生物测定试验中均能诱导植物生长。
T3383 Cimifugin

升麻素,Cimitin

Others Others
Cimifugin (Cimitin) 是中草药Saposhnikovia divaricate 的一种生物活性成分。它能够调节紧密连接减少上皮衍生的主动关键因子,对过敏性炎症产生抑制作用。
TMA0955 Thunberginol C

Antifection Microbiology/Virology
Thunberginol C exhibits antimicrobial activity against oral bacteria. It shows antiallergic activity in the in vitro bioassay using the Schults-Dale reaction in sensitized guinea pig bronchial muscle.
TN2552 1-Methyl-2-nonylquinolin-4(1H)-one

Others Others
1-Methyl-2-nonylquinolin-4(1H)-one has anti-inflammatory activity, it exhibits inhibitory activity on leukotriene biosynthesis in a bioassay using human polymorphonuclear granulocytes, with IC50 values of 12.1 microM.
TN4475 Macrocarpal C

ROS; Antifection Immunology/Inflammation; Microbiology/Virology
Macrocarpal C, isolated from the fresh leaves of Eucalyptus globulus Labill. (Lan An) and identified as its major antifungal component by bioassay-guided purification, the antifungal action of macrocarpal C was associated with increases of membrane permea

天然产物

3-Methoxyphenylacetic acid
Cat.No: Fr13883
Synonym:
Target: Others
(22S,23S)-Homobrassinolide
Cat.No: T41372
Synonym: 油菜素内酯,SSHB
Target: Others
Cimifugin
Cat.No: T3383
Synonym: 升麻素,Cimitin
Target: Others
Thunberginol C
Cat.No: TMA0955
Synonym:
Target: Antifection
1-Methyl-2-nonylquinolin-4(1H)-one
Cat.No: TN2552
Synonym:
Target: Others
Macrocarpal C
Cat.No: TN4475
Synonym:
Target: ROS, Antifection
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