3
1
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T16348 |
NS5806
NS-5806 |
Potassium Channel | Membrane transporter/Ion channel |
NS5806 是钾电流的激活剂,可增加 KV4.3/KChIP2峰值电流幅度,EC50值为 5.3 μM。它会在包含 KChIP2 的通道复合体中降低 KV4.2 和 KV4.3 电流衰减。 | |||
T9009 |
ICA-105574
ICA,3-nitro-N-[4-phenoxyphenyl]-benzamide |
HER | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
ICA-105574 (ICA) 是 hERG 通道激活剂。它通过消除 hERG 通道的失活从而增强 hERG 通道活性。它可以把电流幅度急剧增加到原来的 10 倍以上,其EC50值为 0.5 +/- 0.1 μM,Hill 斜率 (n(H)) 为 3.3 +/- 0.2。 | |||
T76392 |
β-Bag cell peptide
|
||
β-Bag cell peptide是一种提高袋细胞神经元(bag cell neuron)中cAMP水平、并能降低电压依赖性钾电流的神经活性肽。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T37609 |
(rel)-Asperparaline A
|
||
Aspergillimide is a fungal metabolite originally isolated from A. japonicus.1 It reduces nicotinic acetylcholine receptor (nAChR) peak and slowly-desensitizing amplitudes induced by acetylcholine in silkworm (B. mori) larval neurons (IC50s = 20.2 and 39.6 nM, respectively) but has no effect on chicken α3β4-, α4β2-, and α7-containing nAChRs.2 Dietary administration of aspergillimide A (10 μg/g of diet) induces paralysis in silkworm fourth instar larvae.1 Aspergillimide A (10 and 20 mg/kg) reduces... |