首页 工具
登录
购物车

搜索结果

Search Results for " adenoma "

4

抑制剂 & 化合物

2

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T21294 Polmacoxib

CG-100649,帕马考昔,CG100649,CG 100649

COX; Carbonic Anhydrase Immunology/Inflammation; Metabolism; Neuroscience
Polmacoxib (CG 100649) 是一流的 NSAID 候选药物,是碳酸酐酶 (CA) 和 COX-2 的双重抑制剂。它在小鼠模型中抑制大肠腺瘤和肿瘤生长。
T8359 Lanreotide acetate

Lanreotide acetate (108736-35-2 free base),BIM 23014 (acetate),BIM 23014 acetate

Others Others
Lanreotide acetate (BIM 23014 acetate) 是生长抑素类似物,具有抗肿瘤活性,可用于类癌综合症。
T41179 CL 82198 hydrochloride

CL 82198 hydrochloride is a selective inhibitor of MMP-13 (89% inhibition at 10μg/mL) that displays no activity at MMP-1, MMP-9 or TACE. Inhibitsin vitroinvasion by the human pituitary adenoma cell line HP75. Rescues paclitaxel induced axon degradation and reduces associated neurotoxicity in zebrafish.
T74815 SLC26A3-IN-2

SLC26A3-IN-2 是一种口服有效的阴离子交换蛋白 SLC26A3的抑制剂 (IC50=360 nM)。SLC26A3 属于溶质载体 (SLC) 蛋白,属于 SLC26 家族。SLC26 家族对氯化物、碳酸氢盐、硫酸盐和草酸盐具有广泛的阴离子特异性。SLC26A3 在腺瘤 (DRA) 中下调,参与氯化物和草酸盐的肠道吸收。SLC26A3 功能突变的丧失与氯离子丢失性腹泻有关。

化合物

Polmacoxib
Cat.No: T21294
Synonym: CG-100649,帕马考昔,CG100649,CG 100649
Target: COX, Carbonic Anhydrase
Lanreotide acetate
Cat.No: T8359
Synonym: Lanreotide acetate (108736-35-2 free base),BIM 23014 (acetate),BIM 23014 acetate
Target: Others
CL 82198 hydrochloride
Cat.No: T41179
Synonym:
Target:
SLC26A3-IN-2
Cat.No: T74815
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TQ0193 N2,N2-Dimethylguanosine

N2,N2-二甲基鸟苷

Endogenous Metabolite Metabolism
N2,N2-Dimethylguanosine 是尿核苷,是 tRNA 的初级代谢产物。
T36472 Tetrahydro-11-deoxy Cortisol

Tetrahydro-11-deoxy cortisol (THS) is the primary urinary metabolite of 11-deoxycortisol. Urinary excretion of THS is elevated in patients with 11β-hydroxylase deficiency, a condition resulting from mutations in the cytochrome P450 (CYP) isoform CYP11B1. Urinary levels of THS are also elevated in patients with adrenocortical carcinoma (ACC) and adrenocortical adenoma (ACA) but are higher in patients with ACC compared to ACA.

天然产物

N2,N2-Dimethylguanosine
Cat.No: TQ0193
Synonym: N2,N2-二甲基鸟苷
Target: Endogenous Metabolite
Tetrahydro-11-deoxy Cortisol
Cat.No: T36472
Synonym:
Target:
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼