Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5336 |
Zacopride hydrochloride
|
Potassium Channel; 5-HT Receptor | GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience |
Zacopride hydrochloride 是5-HT3受体拮抗剂 (Ki:0.38 nM),也是5-HT4受体激动剂 (Ki:373 nM),具有抗焦虑作用。它对精神分裂症具有潜在的研究价值。 | |||
T5336L |
Zacopride
Racemic zacopride |
||
Zacopride is a selective agonist of inward rectifier potassium current (I K1) channel, inhibiting ventricular arrhythmias without affecting atrial arrhythmias. |