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Targets Recommended: PLK

2

抑制剂 & 化合物

1

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T21678 3MB-PP1

PLK Cell Cycle/Checkpoint
3MB-PP1是嘌呤类似物,是一种 Polo 样激酶 1 (Plk1) 抑制剂。在表达类似物敏感的 Plk1 等位基因的细胞中,3MB-PP1 通过靶向 Plk1 阻断有丝分裂进程和细胞分裂。3MB-PP1 特异性抑制类似物敏感的 Ssn3 (Cdk8)。3MB-PP1 抑制 Leu93 突变 Zipper-interacting protein kinase(Leu93-ZIPK),IC50为2 μM。3MB-PP1 可用于细胞分裂和白色念珠菌 (Candida albicans) 菌丝形成的研究。
T27554 HS38

HS 38,HS-38

DAPK Apoptosis
HS38 是一种特异性的 ATP 竞争性 DAPK 抑制剂,对 DAPK1、PIM3 和 ZIPK 的 Kds 分别为 300 nM、200 nM 和 280 nM。 HS38 可用于平滑肌相关疾病的研究。

化合物

3MB-PP1
Cat.No: T21678
Synonym:
Target: PLK
HS38
Cat.No: T27554
Synonym: HS 38,HS-38
Target: DAPK
Cat. No. Product Name Species Expression System
TMPY-04385 ZIP Kinase/DAPK3 Protein, Human, Recombinant (GST)

death-associated protein kinase 3,DLK,ZIP,ZIPK

Human Baculovirus Insect Cells
Death-associated protein kinase 3, also known as DAP kinase 3, ZIP-kinase, DAPK3 and ZIPK, is a nucleus and cytoplasm protein which belongs to theprotein kinase superfamily, CAMK Ser/Thr protein kinase family and DAP kinase subfamily. DAPK3 / ZIPK contains oneprotein kinase domain. It is a serine/threonine kinase which acts as a positive regulator of apoptosis. It phosphorylates histone H3 on 'Thr-11' at centromeres during mitosis. DAPK3 / ZIPK is a homodimer or forms heterodimers with AT...

重组蛋白

ZIP Kinase/DAPK3 Protein, Human, Recombinant (GST)
Cat.No: TMPY-04385
Species: Human
Expression System: Baculovirus Insect Cells
TargetMol Loading
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