Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8435 |
YM90K
YM90K hydrochloride,6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-,1,4-二氢-6-(1H-咪唑-1-基)-7-硝基-2,3-喹喔啉二酮单盐酸盐 |
GluR; iGluR | Membrane transporter/Ion channel; Neuroscience |
YM90K (6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-) hydrochloride 是一种选择性的、有效的AMPA 受体拮抗剂,Ki=84 nM。YM90K 抑制海藻酸酯 (Ki 为 2.2 μM) 和 NMDA (Ki 为 37 μM) 受体的效力较低,并具有神经保护活性。 | |||
T29192 |
YM-900
YM90K,YM 900,YM 90K,YM-90K |
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YM-900, an AMPA receptor antagonist and glutamate receptor antagonist, is used potentially for the treatment of stroke. |