Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4595 |
YHO-13177
YHO 13177,YHO13177 |
BCRP | Membrane transporter/Ion channel |
YHO-13177 是高活性乳腺癌耐药蛋白多药转运通道(BCRP)抑制剂,可增强SN-38活性。 | |||
T13365 |
YHO-13351 free base
|
BCRP | Membrane transporter/Ion channel |
YHO-13351 free base 是 YHO-13177 的水溶性前药,YHO-13177 是 BCRP 的抑制剂。 | |||
T13366 |
YHO-13351
|
Epigenetic Reader Domain | Chromatin/Epigenetic |
YHO-13351 is the water-soluble prodrug of YHO-13177, which is a potent and specific BCRP inhibitor. |