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Cat. No. Product Name Target Signaling Pathways
T6916 OICR-9429

OICR 9429

Histone Methyltransferase; JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
OICR-9429 是一个新颖的相互作用的小分子Wdr5-MLL 拮抗剂,IC50是 5 uM,在体外抑制急性髓性白血病细胞。
T8768 MM-102 TFA

HMTase Inhibitor IX TFA

Histone Methyltransferase Chromatin/Epigenetic
MM-102 TFA (HMTase Inhibitor IX TFA) 是一种有效的 WDR5/MLL 相互作用抑制剂,在 WDR5 结合检测中,IC50为 2.4 nM,Ki 小于 1 nM。
T13334 WDR5-IN-1

Others Others
WDR5-IN-1 is a potent and selective inhibitor of WD repeat domain 5 (WDR5) (Kd <0.02 nM), and also inhibits MLL1 histone methyltransferase (HMT) activity (IC50: 2.2 nM).
T12091 MM-589

JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
MM-589 is a potent WD repeat domain 5 (WDR5) inhibitor and mixed lineage leukemia (MLL) protein-protein interaction.
T12091L MM-589 TFA

JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
MM-589 TFA is a potent WD repeat domain 5 (WDR5)inhibitor and mixed lineage leukemia (MLL) protein-protein interaction.
T63763 WDR5-IN-5

WDR5-IN-5 是选择性的、口服具有活力的、靶向 WD 重复结构域 5 (WDR5)WIN 位点的抑制剂。WDR5-IN-5WDR5 表现出高亲和力 (Ki<0.02 nM)。WDR5-IN-5 表现出抗癌细胞增殖作用以及良好的药代动力学特征。

化合物

OICR-9429
Cat.No: T6916
Synonym: OICR 9429
Target: Histone Methyltransferase, JAK
MM-102 TFA
Cat.No: T8768
Synonym: HMTase Inhibitor IX TFA
Target: Histone Methyltransferase
WDR5-IN-1
Cat.No: T13334
Synonym:
Target: Others
MM-589
Cat.No: T12091
Synonym:
Target: JAK
MM-589 TFA
Cat.No: T12091L
Synonym:
Target: JAK
WDR5-IN-5
Cat.No: T63763
Synonym:
Target:
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