Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13278L |
Valecobulin
CKD-516 |
Others | Others |
Valecobulin is a potent β-tubulin polymerization inhibitor. Valecobulin is a valine prodrug of (S516) and an avascular disrupting compound. | |||
T13278 |
Valecobulin hydrochloride
CKD-516 hydrochloride |
Microtubule Associated | Cytoskeletal Signaling |
Valecobulin hydrochloride (CKD-516 hydrochloride) 是 S516 的缬氨酸前体药和血管阻断剂。Valecobulin hydrochloride 对β-微管蛋白聚合有强效的抑制作用,对小鼠和人类的实体肿瘤具有显著的抗肿瘤活性。 |