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Cat. No. Product Name Target Signaling Pathways
T33243 MC-Val-Cit-PAB-VX765

Belnacasan-conjugate,VX765-conjugate,MC-Val-Cit-PABC-VX765

MC-VAL-CIT-PAB-VX765 or MC-VAL-CIT-PABC-VX765 is a VX765 derivative that can be conjugated to antibodies, proteins, or polymers for targeted drug delivery. MC-Val- CIT -PAB is a cathepsin cleavable ADC connector, which has been widely used in the preparat
T6090 Belnacasan

VX-765

Caspase Apoptosis; Proteases/Proteasome
Belnacasan (VX-765) 是一种具有口服活性的 IL 转换酶/caspase-1 抑制剂,是 VRT-043198 的口服生物活性前药,作用于外周血单核细胞,可抑制 LPS 诱导的 IL-1β 和 IL-18 释放。

化合物

MC-Val-Cit-PAB-VX765
Cat.No: T33243
Synonym: Belnacasan-conjugate,VX765-conjugate,MC-Val-Cit-PABC-VX765
Target:
Belnacasan
Cat.No: T6090
Synonym: VX-765
Target: Caspase
TargetMol Loading
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