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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T7897 PK150

Others; Antibacterial Microbiology/Virology; Others
PK150 是一种 Sorafenib 类似物,具有抗菌活性。它抑制甲氧西林敏感金黄色葡萄球菌,耐甲氧西林金黄色葡萄球菌,万古霉素中介金黄色葡萄球菌的 MIC 分别为 0.3,0.3-1,0.3 µM。
TQ0046 Bavisant

JNJ-31001074

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Bavisant (JNJ-31001074) 是一种特异性和口服活性的人 H3 受体拮抗剂。 Bavisant 可用于作用机制的研究,包括觉醒和认知以及 ADHD 的治疗。
T10462L Bavisant dihydrochloride hydrate

JNJ31001074AAC

Others Others
Bavisant dihydrochloride hydrate (JNJ31001074AAC) is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition, with potential as a treatment for ADHD. in vivo: Mean change
T10462 Bavisant dihydrochloride

Others Others
Bavisant (JNJ-310010740) dihydrochloride is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition.
T74776 Antibacterial agent 139

Antibacterial agent 139 对革兰氏阳性菌具有抗菌活性。Antibacterial agent 139 具有抗 MRSA、抗 VISA 和抗 LRSE 活性。Antibacterial agent 139 去极化细菌细胞膜。
T14359 AVX 13616

Others Others
AVX 13616 shows the potent in vivo antibacterial activity of Avexa’s lead antibacterial candidate; particularly against drug-resistant Staphylococcus pathogens. IC50 value: 2-4 ug/ml (MICs) Target: antibacterial agent AVX13616 was as active as mupirocin i

化合物

PK150
Cat.No: T7897
Synonym:
Target: Others, Antibacterial
Bavisant
Cat.No: TQ0046
Synonym: JNJ-31001074
Target: Histamine Receptor
Bavisant dihydrochloride hydrate
Cat.No: T10462L
Synonym: JNJ31001074AAC
Target: Others
Bavisant dihydrochloride
Cat.No: T10462
Synonym:
Target: Others
Antibacterial agent 139
Cat.No: T74776
Synonym:
Target:
AVX 13616
Cat.No: T14359
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
TN1297 5-O-Methylvisamminol

5-O-甲基维斯阿米醇,5-O-甲维阿斯米醇,5-O-甲基维生素B

Others Others
5-O-Methylvisamminol 是一种在植物界中有限存在的呋喃色酮,提取于青冈草。它是很好的菊科植物化学分类学标记,也可用于化学系统发育。
TQ0240 6"-O-Apiosyl-5-O-Methylvisammioside

Others Others
6”-O-Apiosyl-5-O-Methylvisammioside 是中药颈复康的成分之一,颈复康具有活血通络,散风止痛的作用。
T3413 5-O-Methylvisammioside

5-O-Methylvisamminol glucoside,4'-O-β-D-Glucosyl-5-O-methylvisamminol,5-O-甲基维斯阿米醇苷

Others Others
5-O-Methylvisammioside (4'-O-β-D-Glucosyl-5-O-methylvisamminol) 是一种天然产物,分离自防风。
TN7098 visamminol-3'-O- glucoside

Others Others
visamminol-3'-O- glucoside 是在 Eranthis Salisb 属中检测到 visamminol-3'-O-葡萄糖苷。
TN4542 Methyl-Dodovisate A

Others Others
Methyl-Dodovisate A is a natural product from Dodonaea viscosa.
T80008 Stevisaliosides D

Phosphatase Metabolism
Stevisaliosides D (Compound 5) 是从甜叶菊根中提取的化合物,具有抑制PTP1B的活性(IC50:31.8 μM),应用于抗糖尿病研究。
TN5740 Visartiside E

Visartiside E 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5740,CAS号为 1212005-08-7。
TN6943 visamminol

visamminol is a natural product.
T80007 Stevisalioside A

Phosphatase Metabolism
Stevisalioside A (Compound 2),一种从甜叶菊根提取的化合物,展现出抗糖尿病的口服活性。该化合物有效抑制PTP1B,IC50为526.8 μM,并能降低Stevisalioside A引起的高血糖小鼠血糖水平,改善餐后血糖峰值及口服葡萄糖和胰岛素耐量测试结果。
T83573 (2′S)-4′-O-β-D-apiofuranosyl-(1→6)-O-β-D-glucopyranosylvisamminol

"(2′S)-4′-O-β-D-apiofuranosyl-(1→6)-O-β-D-glucopyranosylvisamminol" 是 Saposhnikovia divaricata 根部提取的一种糖苷,展现了轻度抗肿瘤活性。

天然产物

5-O-Methylvisamminol
Cat.No: TN1297
Synonym: 5-O-甲基维斯阿米醇,5-O-甲维阿斯米醇,5-O-甲基维生素B
Target: Others
6"-O-Apiosyl-5-O-Methylvisammioside
Cat.No: TQ0240
Synonym:
Target: Others
5-O-Methylvisammioside
Cat.No: T3413
Synonym: 5-O-Methylvisamminol glucoside,4'-O-β-D-Glucosyl-5-O-methylvisamminol,5-O-甲基维斯阿米醇苷
Target: Others
visamminol-3'-O- glucoside
Cat.No: TN7098
Synonym:
Target: Others
Methyl-Dodovisate A
Cat.No: TN4542
Synonym:
Target: Others
Stevisaliosides D
Cat.No: T80008
Synonym:
Target: Phosphatase
Visartiside E
Cat.No: TN5740
Synonym:
Target:
visamminol
Cat.No: TN6943
Synonym:
Target:
Stevisalioside A
Cat.No: T80007
Synonym:
Target: Phosphatase
(2′S)-4′-O-β-D-apiofuranosyl-(1→6)-O-β-D-glucopyranosylvisamminol
Cat.No: T83573
Synonym:
Target:
TargetMol Loading
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