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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7897 |
PK150
|
Others; Antibacterial | Microbiology/Virology; Others |
PK150 是一种 Sorafenib 类似物,具有抗菌活性。它抑制甲氧西林敏感金黄色葡萄球菌,耐甲氧西林金黄色葡萄球菌,万古霉素中介金黄色葡萄球菌的 MIC 分别为 0.3,0.3-1,0.3 µM。 | |||
TQ0046 |
Bavisant
JNJ-31001074 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Bavisant (JNJ-31001074) 是一种特异性和口服活性的人 H3 受体拮抗剂。 Bavisant 可用于作用机制的研究,包括觉醒和认知以及 ADHD 的治疗。 | |||
T10462L |
Bavisant dihydrochloride hydrate
JNJ31001074AAC |
Others | Others |
Bavisant dihydrochloride hydrate (JNJ31001074AAC) is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition, with potential as a treatment for ADHD. in vivo: Mean change | |||
T10462 |
Bavisant dihydrochloride
|
Others | Others |
Bavisant (JNJ-310010740) dihydrochloride is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition. | |||
T74776 | Antibacterial agent 139 | ||
Antibacterial agent 139 对革兰氏阳性菌具有抗菌活性。Antibacterial agent 139 具有抗 MRSA、抗 VISA 和抗 LRSE 活性。Antibacterial agent 139 去极化细菌细胞膜。 | |||
T14359 |
AVX 13616
|
Others | Others |
AVX 13616 shows the potent in vivo antibacterial activity of Avexa’s lead antibacterial candidate; particularly against drug-resistant Staphylococcus pathogens. IC50 value: 2-4 ug/ml (MICs) Target: antibacterial agent AVX13616 was as active as mupirocin i |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN1297 |
5-O-Methylvisamminol
5-O-甲基维斯阿米醇,5-O-甲维阿斯米醇,5-O-甲基维生素B |
Others | Others |
5-O-Methylvisamminol 是一种在植物界中有限存在的呋喃色酮,提取于青冈草。它是很好的菊科植物化学分类学标记,也可用于化学系统发育。 | |||
TQ0240 |
6"-O-Apiosyl-5-O-Methylvisammioside
|
Others | Others |
6”-O-Apiosyl-5-O-Methylvisammioside 是中药颈复康的成分之一,颈复康具有活血通络,散风止痛的作用。 | |||
T3413 |
5-O-Methylvisammioside
5-O-Methylvisamminol glucoside,4'-O-β-D-Glucosyl-5-O-methylvisamminol,5-O-甲基维斯阿米醇苷 |
Others | Others |
5-O-Methylvisammioside (4'-O-β-D-Glucosyl-5-O-methylvisamminol) 是一种天然产物,分离自防风。 | |||
TN7098 |
visamminol-3'-O- glucoside
|
Others | Others |
visamminol-3'-O- glucoside 是在 Eranthis Salisb 属中检测到 visamminol-3'-O-葡萄糖苷。 | |||
TN4542 |
Methyl-Dodovisate A
|
Others | Others |
Methyl-Dodovisate A is a natural product from Dodonaea viscosa. | |||
T80008 |
Stevisaliosides D
|
Phosphatase | Metabolism |
Stevisaliosides D (Compound 5) 是从甜叶菊根中提取的化合物,具有抑制PTP1B的活性(IC50:31.8 μM),应用于抗糖尿病研究。 | |||
TN5740 |
Visartiside E
|
||
Visartiside E 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5740,CAS号为 1212005-08-7。 | |||
TN6943 |
visamminol
|
||
visamminol is a natural product. | |||
T80007 |
Stevisalioside A
|
Phosphatase | Metabolism |
Stevisalioside A (Compound 2),一种从甜叶菊根提取的化合物,展现出抗糖尿病的口服活性。该化合物有效抑制PTP1B,IC50为526.8 μM,并能降低Stevisalioside A引起的高血糖小鼠血糖水平,改善餐后血糖峰值及口服葡萄糖和胰岛素耐量测试结果。 | |||
T83573 |
(2′S)-4′-O-β-D-apiofuranosyl-(1→6)-O-β-D-glucopyranosylvisamminol
|
||
"(2′S)-4′-O-β-D-apiofuranosyl-(1→6)-O-β-D-glucopyranosylvisamminol" 是 Saposhnikovia divaricata 根部提取的一种糖苷,展现了轻度抗肿瘤活性。 |