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Cat. No. Product Name Target Signaling Pathways
T14349 Auristatin F

Microtubule Associated Cytoskeletal Signaling
Auristatin F 是一种有效的微管抑制剂和血管损伤剂。 Auristatin F 可用于抗体-药物偶联物。
T13278 Valecobulin hydrochloride

CKD-516 hydrochloride

Microtubule Associated Cytoskeletal Signaling
Valecobulin hydrochloride (CKD-516 hydrochloride) 是 S516 的缬氨酸前体药和血管阻断剂。Valecobulin hydrochloride 对β-微管蛋白聚合有强效的抑制作用,对小鼠和人类的实体肿瘤具有显著的抗肿瘤活性。
T37024 Mca-DEVDAPK(Dnp)-OH

Mca-DEVDAPK(Dnp)-OH 是 caspase-3 的荧光底物。
T2511 Plinabulin

普那布林,NPI-2358

Microtubule Associated Cytoskeletal Signaling
Plinabulin (NPI-2358) 是一种抗微管蛋白解聚肿瘤细胞的血管破坏剂,选择性地靶向并结合到微管蛋白的秋水仙碱结合位点,从而中断微管动力学的平衡。它对人肿瘤细胞系具有抑制作用,对 HT-29 细胞系的IC50值为 9.8 nM。
T68273 BNC105P

BNC105P is a benzofuran-based vascular disrupting agent (VDA) prodrug with potential anti-vascular and antineoplastic activities. Upon administration vascular disrupting agent BNC105P, the disodium phosphate ester of BNC105, is rapidly converted to BNC105; in activated endothelial cells, BNC105 binds to tubulin and inhibits its polymerization, which may result in a blockage of mitotic spindle formation, cell cycle arrest, and disruption of the tumor vasculature. Hypoxic conditions ensue, deprivi...

化合物

Auristatin F
Cat.No: T14349
Synonym:
Target: Microtubule Associated
Valecobulin hydrochloride
Cat.No: T13278
Synonym: CKD-516 hydrochloride
Target: Microtubule Associated
Mca-DEVDAPK(Dnp)-OH
Cat.No: T37024
Synonym:
Target:
Plinabulin
Cat.No: T2511
Synonym: 普那布林,NPI-2358
Target: Microtubule Associated
BNC105P
Cat.No: T68273
Synonym:
Target:
TargetMol Loading
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