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抑制剂 & 化合物

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Cat. No.	Product Name	Target	Signaling Pathways
TP1205	Velmupressin acetate V2 receptor (V2R) agonist,c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate
	c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively.
T15273	Fedovapagon VA483,A106483	Vasopressin Receptor	GPCR/G Protein
	Fedovapagon (VA106483) 是一种具有选择性和高效性的加压素 V2 受体 (V2R) 激动剂，可抑制斑马鱼节间血管的生长。Fedovapagon 可用于研究膀胱过度活动症、夜尿症和膀胱疼痛综合征。
T80198	Vasopressin Dimer (anti-parallel) (TFA)	Vasopressin Receptor	GPCR/G Protein
	Vasopressin Dimer (anti-parallel) TFA为Vasopressin的反平行二聚体形式，能够激活G蛋白偶联受体V1aR、V1bR、V2R和OTR四种。
TP1473	Velmupressin c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2
	c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 is a selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07nM and 0.02 nM for hV2R and rV2R, respectively.
T80197	Vasopressin Dimer (parallel) (TFA)	Vasopressin Receptor	GPCR/G Protein
	Vasopressin Dimer (parallel) TFA为Vasopressin的平行二聚体，能够激活G蛋白偶联受体V1aR、V1bR、V2R及OTR四种。
T64174	Vasopressin V2 receptor antagonist 1
	Vasopressin V2 receptor antagonist 1 (Compound 4g) 是一种 vasopressin V2receptor (V2R) 拮抗剂 (Ki: 3.8 nM)。Vasopressin V2 receptor antagonist 1 可以用于研究常染色体显性多囊肾病 (ADPKD)。
TP1560	c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm
	c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm a highly efficient, selective and short-acting peptide V2 receptor agonist (V2R), with EC50s of hV2R and rV2R being 0.25 and 0.05 nM, respectively.
T80138	(D-Arg8)-Inotocin	Vasopressin Receptor	GPCR/G Protein
	"(D-Arg8)-Inotocin"是一种对加压素受体V1aR表现出高效、选择性和竞争性拮抗作用的化合物，其Ki值为1.3 nM。该化合物对人类V1aR具有显著的选择性，相较于其他三种亚型(OTR, V1bR, V2R)，其选择性超过3000倍。

化合物

Velmupressin acetate

Cat.No: TP1205

Synonym: V2 receptor (V2R) agonist,c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate

Target:

Fedovapagon

Cat.No: T15273

Synonym: VA483,A106483

Target: Vasopressin Receptor

Vasopressin Dimer (anti-parallel) (TFA)

Cat.No: T80198

Synonym:

Target: Vasopressin Receptor

Velmupressin

Cat.No: TP1473

Synonym: c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2

Target:

Vasopressin Dimer (parallel) (TFA)

Cat.No: T80197

Synonym:

Target: Vasopressin Receptor

Vasopressin V2 receptor antagonist 1

Cat.No: T64174

Synonym:

Target:

c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm

Target: Vasopressin Receptor

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPH-03132	AVPR2 Protein, Pig, Recombinant (His & SUMO) AVPR2,Vasopressin V2 receptor,V2R,AVPR V2,Antidiure...	Sus scrofa (Pig)	E. coli
	Receptor for arginine vasopressin. The activity of this receptor is mediated by G proteins which activate adenylate cyclase. Involved in renal water reabsorption. AVPR2 Protein, Pig, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 24.7 kDa and the accession number is P32307.