Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP2105L |
UFP-101 acetate
UFP-101 acetate(849024-68-6 free base) |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
UFP-101 acetate 是一种特异性和竞争性 NOP 受体拮抗剂 (pKi = 10.24),其特异性是 δ、μ 和 κ 阿片受体的 3000 倍以上。 | |||
TP2105 |
UFP-101
|
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Potent, selective and competitive silent antagonist for the NOP opioid receptor. Binds to NOP with high affinity (pKi = 10.24) and displays > 3000-fold selectivity over δ, μ and κ opioid receptors. Antinociceptive and opposes the action of nociceptin in v |