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Cat. No. Product Name Target Signaling Pathways
T61472 Tubulin inhibitor 18

Tubulin inhibitor 18 (compound 5j) is a highly potent chalcone compound that effectively inhibits tubulin. Its unique molecular structure renders Tubulin inhibitor 18 as a promising candidate for cancer research [1].
T17181 TVB-3664

Fatty Acid Synthase Metabolism
TVB-3664 是一种具有口服具有活力的、选择性的、可逆的、具有高生物利用度的脂肪酸合酶抑制剂,其对人和老鼠棕榈酸酯合成的IC50分别为 18 nM 和 12 nM。可显著抑制微管蛋白棕榈酰化和 mRNA 表达。
T62477 Tubulin polymerization-IN-18

Tubulin aggregation-IN-18 (compound 3) 是一种有效的 tubulin 聚合抑制剂,具有潜力进行乳腺癌和耐药结肠癌的研究。
T36856 UA 62784

Inhibitor of microtubule polymerization in vitro. Interacts with tubulin dimers and promotes the accumulation of mammalian cells in apoptosis. Potentiates antiproliferative effects of vinblastine in H2B-GFP HeLa cells. Originally thought to inhibit CENP-E ATPase activity. Tcherniuk et al (2011) UA62784 is a cytotoxic inhibitor of microtubules, not CENP-E. Chem.Biol. 18 631 PMID:21609844 |Maiato and Logarinho et al (2011) Motor-dependent and -independent roles of CENP-E at kinetochores: the cauti...

化合物

Tubulin inhibitor 18
Cat.No: T61472
Synonym:
Target:
TVB-3664
Cat.No: T17181
Synonym:
Target: Fatty Acid Synthase
Tubulin polymerization-IN-18
Cat.No: T62477
Synonym:
Target:
UA 62784
Cat.No: T36856
Synonym:
Target:
TargetMol Loading
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