Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T34206 |
Pyroglutaminyl-seryl-leucinamide
Thyrotropin releasing hormone-AN,Trh-AN,Pyr-ser-leu-NH2 |
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Pyroglutaminyl-seryl-leucinamide is a bioactive chemical. | |||
T13072 |
Taltirelin acetate
TA-0910 acetate |
Thyroid hormone receptor(THR) | Endocrinology/Hormones |
Taltirelin acetate (TA-0910 acetate) 是促甲状腺激素释放激素受体(TRH-R)超激动剂(IC50:910 nM),能够刺激细胞溶质Ca2+浓度增加 (Ca2+释放) ,其EC50值为 36 nM。 | |||
T33438 |
MK771
MK-771,MK 771 |
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MK771 is a therapeutic agent and an analog of the Thyrotropin Releasing Hormone (TRH). TRH and its analogs may be useful in combating some of the withdrawal symptoms in opiate-dependent subjects. | |||
T7590 |
Taltirelin
TA-0910,他替瑞林 |
Thyroid hormone receptor(THR) | Endocrinology/Hormones |
Taltirelin (TA-0910) 是促甲状腺激素释放激素受体(TRH-R)超激动剂(IC50:910 nM),能够刺激细胞溶质 Ca2+浓度增加 (Ca2+释放) (EC50:36 nM)。 | |||
T75850 |
JKC363 TFA
|
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JKC363 TFA为选择性MC4受体拮抗剂,MC4受体(IC50=0.5 nM)亲和力是MC3受体(44.9 nM)的90倍。JKC363 TFA能阻断α-MSH对TRH释放的刺激,显示出抗痛觉效果。 | |||
TMIH-0550 |
Taltirelin-13C-d3
|
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Taltirelin-13C-d3 是 Taltirelin 的 13C 和氘代化合物。Taltirelin 的 CAS 号为 103300-74-9。Taltirelin 是促甲状腺激素释放激素受体(TRH-R)超激动剂(IC50:910 nM),能够刺激细胞溶质Ca2+浓度增加 (Ca2+释放) (EC50:36 nM)。 |