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Cat. No. Product Name Target Signaling Pathways
T0080 Trapidil

唑嘧胺,乐可安,Rocornal,Trapymine,Avantrin,Trapymin,AR-12008

PDGFR; PDE Angiogenesis; Metabolism; Tyrosine Kinase/Adaptors
Trapidil (Avantrin) 是一种抗血小板药物,是一种血管扩张剂,有特异性血小板衍生生长因子。
T67498 3-Amino-1,2,4-triazole

Amitrole,3-AT,1H-1,2,4-Triazol-5-amine,Trapidil impurity B

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
3-Amino-1,2,4-triazole (Trapidil impurity B) 是一种过氧化氢酶抑制剂,能够诱导过氧化氢解毒的补偿机制。 该机制涉及增加谷胱甘肽过氧化物酶和谷胱甘肽还原酶的活性。
T30110 AR 12456

AR12456,AR-12456

AR-12456 is a Trapidil derivative that prevents serum hyperlipidemia in guinea pigs.
T30111 AR 12465

AR-12465

AR 12465 is a trapidil derivative which may affect LDL receptor mediated uptake and degradation of 125 I-LDL by human skin fibroblasts (HSF) and human hepatic cells (HEP G2).

化合物

Trapidil
Cat.No: T0080
Synonym: 唑嘧胺,乐可安,Rocornal,Trapymine,Avantrin,Trapymin,AR-12008
Target: PDGFR, PDE
3-Amino-1,2,4-triazole
Cat.No: T67498
Synonym: Amitrole,3-AT,1H-1,2,4-Triazol-5-amine,Trapidil impurity B
Target: Reactive Oxygen Species
AR 12456
Cat.No: T30110
Synonym: AR12456,AR-12456
Target:
AR 12465
Cat.No: T30111
Synonym: AR-12465
Target:
TargetMol Loading
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