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Cat. No. Product Name Target Signaling Pathways
T6345 Tirbanibulin

KX2-391,KX-01

Microtubule Associated; Src Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Tirbanibulin (KX2-391) 是一种高度选择性的 Src 激酶抑制,靶向 Src 的多肽底物结合位点,对多种癌症有疗效。
T15675 Tirbanibulin Mesylate

KX2-391 Mesylate,KX01 Mesylate

Microtubule Associated; Src Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Tirbanibulin Mesylate (KX01 Mesylate) 是一种 Src 抑制剂,靶向 Src 的肽底物位点。在肿瘤细胞中,GI50值为 9-60 nM。
T15674 Tirbanibulin dihydrochloride

KX-01 (dihydrochloride),KX2-391 (dihydrochloride)

Src Angiogenesis; Tyrosine Kinase/Adaptors
Tirbanibulin is an inhibitor of Src that targets the peptide substrate site of Src (GI50: 9-60 nM in cancer cell lines).

化合物

Tirbanibulin
Cat.No: T6345
Synonym: KX2-391,KX-01
Target: Microtubule Associated, Src
Tirbanibulin Mesylate
Cat.No: T15675
Synonym: KX2-391 Mesylate,KX01 Mesylate
Target: Microtubule Associated, Src
Tirbanibulin dihydrochloride
Cat.No: T15674
Synonym: KX-01 (dihydrochloride),KX2-391 (dihydrochloride)
Target: Src
TargetMol Loading
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