Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15674 |
Tirbanibulin dihydrochloride
KX-01 (dihydrochloride),KX2-391 (dihydrochloride) |
Src | Angiogenesis; Tyrosine Kinase/Adaptors |
Tirbanibulin is an inhibitor of Src that targets the peptide substrate site of Src (GI50: 9-60 nM in cancer cell lines). | |||
T6345 |
Tirbanibulin
KX2-391,KX-01 |
Microtubule Associated; Src | Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors |
Tirbanibulin (KX2-391) 是一种高度选择性的 Src 激酶抑制,靶向 Src 的多肽底物结合位点,对多种癌症有疗效。 | |||
T15675 |
Tirbanibulin Mesylate
KX2-391 Mesylate,KX01 Mesylate |
Microtubule Associated; Src | Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors |
Tirbanibulin Mesylate (KX01 Mesylate) 是一种 Src 抑制剂,靶向 Src 的肽底物位点。在肿瘤细胞中,GI50值为 9-60 nM。 |