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Cat. No.	Product Name	Target	Signaling Pathways
T7693	Thiorphan	Neprilysin	Metabolism
	Thiorphan 是选择性neprilysin 抑制剂 (IC50:6.9 nM) 。
T25676	Leucine thiorphan Leu-thiorphan
	Leucine thiorphan is an inhibitor of enkephalinase.
T71161	Thiorphan disulfide
	Thiorphan disulfide is an impurity of Racecadotril -- an antidiarrheal and enkephalinase inhibitor that reduces the amount of water and electrolytes absorbed into the intestine.
T68601	Azidothiorphan
	Azidothiorphan is a photoaffinity ligand for the active site of the neutral endopeptidase 24.11. After ultraviolet irradiation the inhibitor binds irreversibly to the enzyme, and photolabeling occurs at the active site. The competitive inhibitor thiorphan protects the endopeptidase from inactivation.
T1176	Racecadotril Acetorphan,消旋卡多曲	Neprilysin; Proteasome	Metabolism; Proteases/Proteasome; Ubiquitination
	Racecadotril (Acetorphan) 是一种中性内肽酶 (NEP) 抑制剂，具有止泻作用。Racecadotril 及其活性代谢物 Thiorphan 抑制小鼠脑中纯化的NEP 活性，Ki 分别为 4500 和 6.1 nM。
T25316	Dexecadotril Retorphan
	Dexecadotril is a powerful and selective neprilysin inhibitor. It behaves as a prodrug of the enantiomer of thiorphan.
T71145	Racecadotril-d5
	Racecadotril-d5 is intended for use as an internal standard for the quantification of racecadotril by GC- or LC-MS. Racecadotril is a prodrug form of the neprilysin (NEP) inhibitor thiorphan. In vivo, racecadotril reduces or prevents castor oil-induced diarrhea without delaying intestinal transit in rats when administered at doses of 80 or 100 mg/kg, respectively. It also decreases the duration of diarrhea and increases body weight gain in a neonatal gnotobiotic pig model of human rotavirus-indu...

化合物

Cat.No: T7693

Target: Neprilysin

Leucine thiorphan

Cat.No: T25676

Synonym: Leu-thiorphan

Thiorphan disulfide

Cat.No: T71161

Cat.No: T68601

Cat.No: T1176

Synonym: Acetorphan,消旋卡多曲

Target: Neprilysin, Proteasome

Cat.No: T25316

Synonym: Retorphan

Racecadotril-d5

Cat.No: T71145

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