Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7753 |
Thalidomide-O-COOH
Cereblon ligand 3,E3 ligase Ligand 3,TCE35031 |
Others; Ligand for E3 Ligase | Others; PROTAC |
Thalidomide-O-COOH (Cereblon ligand 3) 是一种基于 Thalidomide 的 Cereblon 配体,可用于募集 CRBN 蛋白。它能够利用 linker 与靶蛋白配体连接,得到 PROTAC 分子。 | |||
T39644 |
Thalidomide-O-C6-COOH
Thalidomide-O-C6-COOH |
||
Thalidomide-O-C6-COOH is a synthetic conjugate comprising an E3 ligase ligand-linker, which combines the Thalidomide derived cereblon ligand with a PROTAC technology linker. | |||
T39643 |
Thalidomide-O-C4-COOH
Thalidomide-O-C4-COOH |
||
Thalidomide-O-C4-COOH is a synthetic conjugate compound, serving as an E3 ligase ligand-linker, which combines a cereblon ligand derived from Thalidomide and a linker utilized in PROTAC technology. | |||
T17914 |
Thalidomide-O-amido-C3-COOH
Cereblon Ligand-Linker Conjugates 7,E3 ligase Ligand-Linker Conjugates 15 |
Others | Others |
Thalidomide-O-amido-C3-COOH is a synthesized conjugate of an E3 ligase ligand-linker compound that combines a cereblon ligand derived from Thalidomide with a linker commonly employed in PROTAC technology. | |||
T40013 |
Thalidomide-O-CH2CONH-CH2COOH
|
Others | Others |
Thalidomide-O-CH2CONH-CH2COOH 是一种合成的 E3 连接酶配体-接头偶联物,它结合了 PROTAC 技术中使用的基于 Thalidomide 的 CRBN 配体和接头。 | |||
T77918 |
Thalidomide-O-C8-COOH
|
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Thalidomide-O-C8-COOH,一种Thalidomide衍生的Cereblon配体,能有效募集CRBN蛋白。通过linker,Thalidomide-O-C8-COOH可与靶蛋白配体结合,构建PROTAC分子。 |