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Cat. No. Product Name Target Signaling Pathways
T1198 Tetracaine hydrochloride

盐酸丁卡因,Amethocaine hydrochloride,Amethocalne HCl,Tetracaine HCl

Calcium Channel; Sodium Channel Membrane transporter/Ion channel; Metabolism
Tetracaine hydrochloride (Amethocalne HCl) 是一种钙通道蛋白抑制剂,可阻断肌浆网中 Ca2+的电压敏感释放。它主要用作眼科的止痒剂和局部用药,可用于表面和脊髓麻醉。
T19644 Benzonatate

Sodium Channel Membrane transporter/Ion channel
Benzonatate 是外周口服镇咳药,对咳嗽延伸受体 (cough stretch receptors) 的活性具有抑制作用。它是丁卡因样代谢物,能够阻断呼吸延伸受体的钠通道并产生局部麻醉作用。
T83095 Anticancer agent 101

Anticanceragent 101,一种丁卡因衍生物,展现出抗癌活性。
T74767 Anticancer agent 102

Anticancer agent 102 是丁卡因的衍生物。Anticancer agent 102 具有抗癌活性. Anticancer agent 102 诱导细胞凋亡。
T72441 Anticancer agent 100

Anticancer agent 100 是一种丁卡因衍生物,具有抗癌活性,可用于癌症研究。
T70538 PD-85639

PD-85639 is a voltage-gated sodium (Na+) channel blocker (75% in 10 min & >95% in 25 min blockage of Na+ current by 25 μM PD85,639; whole-cell patch clamp using primary rat brain neurons) that is shown to target rat brain Nav1.2 with simultaneous high- and low-affinity modes of binding (EC50 = 56 nM/40% & 20 μM/60% at pH 9.0, 5 nM/28% & 3 μM/72% at pH 7.4, against 2 nM [3H]-PD85,639 for binding rat brain synaptosomes; EC50 = 17 nM/39% & 10 μM/61% using at pH 9.0 using rat brain synaptosome membr...

化合物

Tetracaine hydrochloride
Cat.No: T1198
Synonym: 盐酸丁卡因,Amethocaine hydrochloride,Amethocalne HCl,Tetracaine HCl
Target: Calcium Channel, Sodium Channel
Benzonatate
Cat.No: T19644
Synonym:
Target: Sodium Channel
Anticancer agent 101
Cat.No: T83095
Synonym:
Target:
Anticancer agent 102
Cat.No: T74767
Synonym:
Target:
Anticancer agent 100
Cat.No: T72441
Synonym:
Target:
PD-85639
Cat.No: T70538
Synonym:
Target:
TargetMol Loading
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