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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T1167 Cyproterone acetate

Androcur,醋酸环丙氯地孕酮,Cyproterone 17-O-acetate,醋酸环丙孕酮

Androgen Receptor Endocrinology/Hormones
Cyproterone acetate (Cyproterone 17-O-acetate) 是能够抗雄激素(IC50=7.1 nM) 和孕激素合成的类固醇。它与 progesteron 和糖皮质激素受体有亲和力。
T76048 TAK-683 acetate

TAK-683 acetate是一种高效的KISS1R激动剂(IC50=170 pM),改善了代谢稳定性。作为九肽metastin的类似物,对人和大鼠的EC50值分别为0.96 nM和1.6 nM。该化合物通过消耗下丘脑GnRH,能够降低血浆FSH、LH、睾酮水平,展示了对研究激素依赖性前列腺癌的潜力。
T68701 Abarelix acetate

Abarelix acetate is a synthetic third generation gonadotropin-releasing hormone receptor (GnRHR) antagonist. It increases histamine release from rat peritoneal mast cells in vitro and from a human skin model ex vivo. In vivo, abarelix decreases plasma luteinizing hormone (LH) levels six hours post-treatment in castrated rats, with levels returning to baseline within 24 hours.3 Abarelix (2 mg/kg) also transiently decreases plasma testosterone levels in intact rats, with levels returning to baseli...

化合物

Cyproterone acetate
Cat.No: T1167
Synonym: Androcur,醋酸环丙氯地孕酮,Cyproterone 17-O-acetate,醋酸环丙孕酮
Target: Androgen Receptor
TAK-683 acetate
Cat.No: T76048
Synonym:
Target:
Abarelix acetate
Cat.No: T68701
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TC0025 Testosterone acetate

NSC523836,NSC-523836,NSC 523836,醋酸睾酮

Others Others
Testosterone acetate (NSC-523836) 是一种 Testosterone 前药,是一种天然存在的雄激素睾酮酯。它可用于阳痿、虚弱、疲劳和性腺机能减退的研究。
T20976 Clostebol acetate

Clostebolacetate,Clostene,Alfa-Trofodermin,4-CLTA

Clostebol acetate is a synthetic anabolic-androgenic steroid (AAS) and a derivative of testosterone. It acts as a prodrug of clostebol in the body.

天然产物

Testosterone acetate
Cat.No: TC0025
Synonym: NSC523836,NSC-523836,NSC 523836,醋酸睾酮
Target: Others
Clostebol acetate
Cat.No: T20976
Synonym: Clostebolacetate,Clostene,Alfa-Trofodermin,4-CLTA
Target:
TargetMol Loading
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