Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TQ0315 |
Tandospirone
坦度螺酮,SM-3997 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Tandospirone (SM-3997) is a selective partial agonist of 5-HT1A receptor (Ki: 27 nM) that displays selectivity over SR-2, SR-1C, α1, α2, D1 and D2 receptors (Kis: 1300-41000 nM). | |||
T7412 |
Tandospirone citrate
SM-3997 citrate,坦度螺酮柠檬酸盐,枸橼酸坦度螺酮 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Tandospirone citrate (SM-3997 citrate) 是一种选择性5-HT1A 受体激动剂,Ki 为27 nM。 | |||
T62215 | Tandospirone hydrochloride | ||
Tandospirone (SM-3997) hydrochloride 是一种高效的、选择性的 5-HT1A 受体部分激动剂 (Ki: 27 nM),表现出抗焦虑和抗抑郁活性。Tandospirone hydrochloride 能够用于研究中枢神经系统疾病及其潜在机制。 |