Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4257 |
Belizatinib
TSR-011 |
Trk receptor; ALK | Angiogenesis; Tyrosine Kinase/Adaptors |
Belizatinib (TSR-011) 是可口服的ALK 和 TRKA、TRKB、TRKC 双重抑制剂,对野生型重组 ALK 的IC50值为0.7 nM。 | |||
T29020 |
TSR-011-isomer
TSR011 isomer,TSR-011 isomer,Belizatinib isomer |
||
TSR011-isomer, a TrKA/ALK inhibitor, is used potentially for the treatment of solid tumours and lymphoma. |