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Cat. No. Product Name Target Signaling Pathways
T80971 TNIK-IN-6

TNIK-IN-6 (Compound 9) 是一种Traf2和Nck相互作用激酶(TNIK)的抑制剂,具有0.93 nM的IC50,对神经与精神疾病具有重要影响。
T36016 PF 06260933 dihydrochloride

MAP4K4 (HGK) inhibitor (IC50 = 140 nM). Also inhibits MINK and TNIK (IC50 values are 8 and 13 nM, respectively). Improves fasting hyperglycemia in mice. Orally active. Ammirati et al (2015) Discovery of an in vivo tool to establish proof-of-concept for MAP4K4-based antidiabetic treatment. ACS Med.Chem.Lett. 6 1128 PMID:26617966

化合物

TNIK-IN-6
Cat.No: T80971
Synonym:
Target:
PF 06260933 dihydrochloride
Cat.No: T36016
Synonym:
Target:
TargetMol Loading
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