Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7079 |
Batefenterol
GSK961081,TD-5959 |
Adrenergic Receptor; AChR | GPCR/G Protein; Neuroscience |
Batefenterol (TD-5959) 是一种毒蕈碱受体拮抗剂和β2-肾上腺素受体激动剂,对 hM2、hM3和β2-肾上腺素受体有高亲和力,Ki 值分别为 1.4、1.3 和 3.7 nM。 | |||
T68272 |
Batefenterol Succinate
|
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Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties. |