Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11216 |
Eplivanserin (mixture)
Eplivanserin mixture,SR-46349 (mixture) |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist, | |||
T27277 |
Eplivanserin hemifumarate
Eplivanserin,SR46349,Eplivanserin fumarate,SR-46349 Fumarate,SR-46349,SR 46349 |
||
Eplivanserin is an inverse agonist of 5-HT2A. | |||
T11217 |
Eplivanserin
依利色林,SR-46349 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Eplivanserin (SR-46349) 是一种有效和特异性的 5-HT2A 受体拮抗剂,Kd 值为 1.14 nM,在大鼠皮质膜中 IC50 值为 5.8 nM。 |