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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T68781 | 3Ac-SL0101 | ||
3Ac-SL0101 is a potent RSK-specific inhibitor. It facilitates the development of RSK inhibitors as anti-cancer chemotherapeutic agents. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T16896 |
SL 0101-1
SL0101 |
S6 Kinase | MAPK; PI3K/Akt/mTOR signaling |
SL 0101-1 (SL0101) 是一种可透过细胞膜且具有选择性、高效性、可逆性、ATP竞争性的 p90核糖体S6激酶(RSK) 的抑制剂,对 RSK 的 IC50 值为 89 nM。SL 0101-1 (SL0101) 也是一种有效的 RSK1/2 抑制剂,其 Ki 值为 1 μM。 |