Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13887 |
SJF620
|
Others; PROTACs | Others; PROTAC |
SJF620 is a potent degrader of PROTAC BTK(DC50 : 7.9 nM). | |||
T74002 | SJF620 hydrochloride | PROTACs | PROTAC |
SJF620 hydrochloride,作为一种连接Cereblon配体和Btk配体的PROTAC,具备DC50值为7.9 nM。该化合物含Lenalidomide类似物,能有效募集CRBN。 |