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3

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T4176 rac-BHFF

(R,S)-BHFF

GABA Receptor Membrane transporter/Ion channel; Neuroscience
rac-BHFF ((R,S)-BHFF) 是具有口服活性的 GABAB 受体的异构增强剂,有抗焦虑活性。
T34492 Salinazid

Nilazid,Salicylaldehyde isonicotinoyl hydrazone,Salizid,Salizide,Nupasal,SIH1

Others Others
Salinazid (Salicylaldehyde isonicotinoyl hydrazone) 是一种有效的抗结核药。
T61198 FAAH/MAGL-IN-1

FAAH/MAGL-IN-1, also known as compound SIH 3, is a highly effective inhibitor of FAAH (fatty acid amide hydrolase) and MAGL (monoacylglycerol lipase). It exhibits IC50 values of 31 nM and 29 nM against FAAH and MAGL, respectively. This compound shows promising potential for advancing research in the field of neuropathic pain [1].

化合物

rac-BHFF
Cat.No: T4176
Synonym: (R,S)-BHFF
Target: GABA Receptor
Salinazid
Cat.No: T34492
Synonym: Nilazid,Salicylaldehyde isonicotinoyl hydrazone,Salizid,Salizide,Nupasal,SIH1
Target: Others
FAAH/MAGL-IN-1
Cat.No: T61198
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T16340 Nosiheptide

RP 9671,Multhiomycin,那西肽

Antibacterial; Antibiotic Microbiology/Virology
Nosiheptide (Multhiomycin) 是一种由 Streptomyces actuosus 生产的硫肽类抗生素,已被广泛用作动物生长的饲料添加剂。它抑制细菌蛋白质合成,并在特征性大环核心上带有独特的吲哚侧环系统和区域特异性羟基。

天然产物

Nosiheptide
Cat.No: T16340
Synonym: RP 9671,Multhiomycin,那西肽
Target: Antibacterial, Antibiotic
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