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Cat. No. Product Name Target Signaling Pathways
T11213 Epertinib hydrochloride

S-22611 hydrochloride

EGFR; HER Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Epertinib hydrochloride (S-22611 hydrochloride) 是口服可逆的选择性EGFR、HER2和HER4抑制剂,IC50值分别为 1.48、7.15 和 2.49 nM,具有抗肿瘤活性。
T11213L Epertinib

S-22611

EGFR; HER Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Epertinib is a reversible and selective tyrosine kinase inhibitor of EGFR, HER2, and HER4 (IC50s: 1.48 nM, 7.15 nM, and 2.49 nM). It displays a strong antitumor activity.

化合物

Epertinib hydrochloride
Cat.No: T11213
Synonym: S-22611 hydrochloride
Target: EGFR, HER
Epertinib
Cat.No: T11213L
Synonym: S-22611
Target: EGFR, HER
TargetMol Loading
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