Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12738L |
Rivanicline
RJR-2403,(E)-Metanicotine |
Others | Others |
Rivanicline is a neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki=26 nM). It show > 1,000 fold selectivity than α7 receptors(Ki= 36000 nM and IC50 : 26 nM). | |||
T12738L1 |
Rivanicline 2HCl
Rivanicline 2HCl(15585-43-0 Free base) |
AChR | Neuroscience |
Rivanicline 2HCl 是一种选择性神经元烟碱受体(neuronal nicotinic receptor) 的抑制剂,对α4β2 亚型的亲和力较高。 | |||
T68891 |
Rivanicline galactarate
|
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Rivanicline galactarate is a Nicotinic Receptor Agonist that may be useful in the treatment of Ulcerative Colitis. | |||
T12738 |
Rivanicline hemioxalate
RJR-2403 hemioxalate,(E)-Metanicotine hemioxalate |
Others | Others |
Rivanicline hemioxalate (RJR-2403 hemioxalate; (E)-Metanicotine hemioxalate) 是一种神经元烟碱受体 (neuronal nicotinic receptor) 激动剂,对 α4β2 亚型有高度选择性(Ki= 26 nM),比对于 α7 受体的选择性高1000倍(Ki=3.6 μM)。 | |||
T12739 |
Rivanicline oxalate
RJR-2403 oxalate,(E)-Metanicotine oxalate |
Others | Others |
Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM). | |||
T26096 |
RJR-2403 oxalate
RJR 2403 oxalate,Rivanicline oxalate,TC-2403,Metanicotine |
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RJR-2403 oxalate is a highly selective agonist of α4β2 subtype nicotinic receptor. |