Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5S0384 |
Rhapontin
Ponticin,土大黄苷,Rhaponiticin,Rhaponticin,Rhapontigenin glucoside |
Apoptosis; Others | Apoptosis; Others |
Rhapontin (Ponticin) 是药用大黄的一种成分,可减轻KK/Ay 糖尿病小鼠肝脏脂肪变性,改善血糖和血脂,表明其具有显着的降糖作用,有望成为治疗2型糖尿病及其并发症的新药。 | |||
TN2153 |
Rhaponticin 6′′-O-gallate
土大黄苷 6''-O-没食子酸酯,Rhaponticin 6''-O-gallate |
Others | Others |
Rhaponticin 6''-O-gallate showed inhibitory activity of NO production in lipopolysaccharide-activated macrophages, (IC50 = 11-69 microM). | |||
TN2152 |
Rhaponticin 2′′-O-gallate
土大黄苷 2''-O-没食子酸酯,Rhaponticin 2''-O-gallate |
Others | Others |
Rhaponticin 2''-O-gallate showed inhibitory activity of NO production in lipopolysaccharide-activated macrophages, (IC50 = 11-69 microM). | |||
TJS0387 |
Desoxyrhaponticin
去氧土大黄苷,Deoxyrhapontin,脱氧土大黄苷,Deoxyrhaponticin |
Apoptosis; Fatty Acid Synthase | Apoptosis; Metabolism |
Desoxyrhaponticin (Deoxyrhaponticin) 是来自西藏营养食品唐古特大黄中的一种二苯乙烯苷。它是脂肪酸合成酶抑制剂,抑制细胞内 FAS 活性,下调人乳腺癌 MCF-7细胞中 FAS 的表达。它是控制糖尿病餐后高血糖的潜在药物。 |