Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12778L |
RTI-13951-33
|
GPR | Endocrinology/Hormones; GPCR/G Protein |
RTI-13951-33 is an effective and brain-penetrant GPR88 agonist (EC50: 25 nM, in GPR88 cAMP functional assay). | |||
T12778 |
RTI-13951-33 hydrochloride
RTI-13951-33 hydrochloride (2244884-08-8 free base) |
Others | Others |
RTI-13951-33 hydrochloride 是一种有效的、选择性的、可透过血脑屏障的GPR88激动剂。RTI-13951-33 hydrochloride 在 GPR88 cAMP 功能性测定中,EC50值为 25 nM。RTI-13951-33 hydrochloride 可以降低大鼠酒精强化和摄入行为。 |