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Cat. No. Product Name Target Signaling Pathways
T12727 RIP2 kinase inhibitor 1

Others Others
RIP2 kinase inhibitor 1 is a potent and selective receptor interacting inhibitor of protein 2 (RIP2) kinase(RIP2 FP with an IC50 of 0.03 μM ),and is used for autoinflammatory disorders.
T12728 RIP2 Kinase Inhibitor 3

Others; RIP kinase Apoptosis; NF-κB; Others
RIP2 Kinase Inhibitor 3 是一种有效的选择性 受体相互作用蛋白2 激酶抑制剂,IC50 为 1 nM。
T5401 GSK2983559 active metabolite

GSK2983559,RIPK2 inhibitor 1,RIPK2-IN-1

RIP kinase Apoptosis; NF-κB
GSK2983559 active metabolite (RIPK2-IN-1) 是一种受体相互作用蛋白-2 激酶抑制剂。
T74572 RIPK2-IN-2

RIPK2-IN-2 (example 25) 是RIP2 激酶PROTAC 抑制剂。RIPK2-IN-2 可以阻断 RIP2 依赖的促炎信号,调节 RIP2 激酶在自身炎性疾病中的活性。
T36243 PROTAC RIPK degrader-6

PROTACs PROTAC
PROTAC RIPK degrader-6 (example 1) is a PROTAC designed for the targeted degradation of RIP Kinase, featuring a RIP2 kinase inhibitor connected through a linker to a cereblon binder[1].

化合物

RIP2 kinase inhibitor 1
Cat.No: T12727
Synonym:
Target: Others
RIP2 Kinase Inhibitor 3
Cat.No: T12728
Synonym:
Target: Others, RIP kinase
GSK2983559 active metabolite
Cat.No: T5401
Synonym: GSK2983559,RIPK2 inhibitor 1,RIPK2-IN-1
Target: RIP kinase
RIPK2-IN-2
Cat.No: T74572
Synonym:
Target:
PROTAC RIPK degrader-6
Cat.No: T36243
Synonym:
Target: PROTACs
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