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Cat. No. Product Name Target Signaling Pathways
T12728 RIP2 Kinase Inhibitor 3

Others; RIP kinase Apoptosis; NF-κB; Others
RIP2 Kinase Inhibitor 3 是一种有效的选择性 受体相互作用蛋白2 激酶抑制剂,IC50 为 1 nM。
T7504 Necrostatin 2 racemate

5-[(7-氯-1H-吲哚-3-基)甲基]-3-甲基-2,4-咪唑烷二酮,Necrostatin-2 racemate

RIP kinase Apoptosis; NF-κB
Necrostatin 2 racemate (Necrostatin-2 racemate) 是一种特异性的RIPK1抑制剂,是一种稳定型 Nec-1。
T9095 Necrostatin-34

2-{[3-cyano-4-(4-methylphenyl)-6-oxo-1,4

RIP kinase Apoptosis; NF-κB
Necrostatin-34 (2-{[3-cyano-4-(4-methylphenyl)-6-oxo-1,4) 是一种 RIPK1 激酶抑制剂,通过在激酶结构域中占据一个独特的结合口袋,将 RIPK1 激酶稳定在非活性构象中。
T16753 RIP2 kinase inhibitor 2

Others Others
RIP2 kinase inhibitor 2 is a receptor-interacting protein-2 kinase inhibitor.
T12727 RIP2 kinase inhibitor 1

Others Others
RIP2 kinase inhibitor 1 is a potent and selective receptor interacting inhibitor of protein 2 (RIP2) kinase(RIP2 FP with an IC50 of 0.03 μM ),and is used for autoinflammatory disorders.
T39574 RIP2 Kinase Inhibitor 4

RIP2 Kinase Inhibitor 4 is a highly potent and selective RIPK2 PROTAC compound that efficiently degrades RIPK2 (with a pIC50 value of 8) and effectively inhibits the release of TNF-α.

化合物

RIP2 Kinase Inhibitor 3
Cat.No: T12728
Synonym:
Target: Others, RIP kinase
Necrostatin 2 racemate
Cat.No: T7504
Synonym: 5-[(7-氯-1H-吲哚-3-基)甲基]-3-甲基-2,4-咪唑烷二酮,Necrostatin-2 racemate
Target: RIP kinase
Necrostatin-34
Cat.No: T9095
Synonym: 2-{[3-cyano-4-(4-methylphenyl)-6-oxo-1,4
Target: RIP kinase
RIP2 kinase inhibitor 2
Cat.No: T16753
Synonym:
Target: Others
RIP2 kinase inhibitor 1
Cat.No: T12727
Synonym:
Target: Others
RIP2 Kinase Inhibitor 4
Cat.No: T39574
Synonym:
Target:
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