Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6274 |
RO4929097
RG-4733 |
Beta Amyloid; Gamma-secretase | Neuroscience; Proteases/Proteasome; Stem Cells |
RO4929097 (RG-4733) 是 γ secretase 抑制剂,IC50=4 nM,能够抑制细胞内 Aβ40 (EC50:14 nM) 的产生和 Notch (EC50:5 nM) 活性。 |