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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T3185 R112

(E)-Elafibranor

Syk Angiogenesis; Tyrosine Kinase/Adaptors
R112 ((E)-Elafibranor) 是ATP 竞争性的 Syk 激酶抑制剂,它能够抑制Syk 激酶活性,Ki=6 nM,IC50=226 nM。
T36577 K-Biotin-W-Histone H2B (108-125) (trifluoroacetate salt)

K-Biotin-W-Histone H2B (108-125) (trifluoroacetate salt)

Histone H2B (108-125) is a peptide fragment of histone H2B that corresponds to amino acid residues 109-126 of the human histone H2B sequence. It contains an N-terminal biotinylated lysine followed by a tryptophan linker. Histone H2B can be modified by addition of an O-linked N-acetylglucosamine (GlcNAc) moiety to the serine residue at position 112, which promotes monoubiquitination of the lysine at position 120.1 Both of these modifications are associated with active transcription. Histone H2B a...

化合物

R112
Cat.No: T3185
Synonym: (E)-Elafibranor
Target: Syk
K-Biotin-W-Histone H2B (108-125) (trifluoroacetate salt)
Cat.No: T36577
Synonym: K-Biotin-W-Histone H2B (108-125) (trifluoroacetate salt)
Target:
Cat. No. Product Name Target Signaling Pathways
TN4838 Pseurotin A

Antifection Microbiology/Virology
Pseurotin A has immunosuppressive activity, it inhibits immunoglobulin E(IgE) production in vitro.It shows a moderate effect against the phytopathogenic bacteria Erwinia carotovora and Pseudomonas syringae, with IC50 values of 220 and 112 microg ml(-1), r

天然产物

Pseurotin A
Cat.No: TN4838
Synonym:
Target: Antifection
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