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Cat. No. Product Name Target Signaling Pathways
T4996 Atosiban

阿托西班,RWJ22164,RW22164

Oxytocin Receptor; Vasopressin Receptor Endocrinology/Hormones; GPCR/G Protein
Atosiban (RW22164) 是一种脱氨基催产素类似物,是一种九肽,也是竞争性的催产素受体拮抗剂。它是一种宫缩抑制剂,可用于自发早产的研究。
T5148 Atosiban acetate

RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164,醋酸阿托西班

Oxytocin Receptor; Vasopressin Receptor Endocrinology/Hormones; GPCR/G Protein
Atosiban acetate (RW22164) 是一种脱氨基催产素类似物,是一种九肽,也是竞争性的催产素受体拮抗剂。它是一种宫缩抑制剂,可用于自发早产的研究。
T28855 SSR126768A

SSR-126768A,SSR 126768A

Oxytocin Receptor Endocrinology/Hormones; GPCR/G Protein
SSR126768A 是一种新型且具有选择性、口服活性和有效性的催产素(OT)受体拮抗剂,对子宫收缩有抑制作用,可用于预防早产。
T70570 Erlosiban

Erlosiban, also known as OBE001, is a novel, orally active nonpeptide oxytocin receptor antagonist under development for the treatment of preterm labor and improvement in embryo implantation and pregnancy rate in assisted reproductive technology (ART).
T70000 Ebopiprant HCl

Ebopiprant, also known as OBE-022, is an Oral and Selective Prostaglandin F 2α Receptor Antagonist as an Effective and Safe Modality for the Treatment of Preterm Labor. OBE022 exhibits potent tocolytic effects on human tissues ex vivo and animal models in vivo without causing the adverse fetal side effects seen with indomethacin.
T73762 11,12-DiHETrE

11,12-DiHETrE,一种细胞色素P450 (P450) 类二十烷素内源性代谢产物,用于早产研究,并可作为区分NAFL(非酒精性脂肪肝)与NASH(非酒精性脂肪性肝炎)的生物标志物。
T76565 PDC31

PDC31 (THG113.31; ILGHXDYK) 是FPProstaglandin Receptor 的变构和非竞争性抑制剂。PDC31是基于D-氨基酸的寡肽,用作平滑肌收缩剂。PDC31 在体内降低子宫收缩的强度和持续时间,可用于早产和原发性痛经 (PD) 的研究。PDC31 还增强人子宫肌层细胞中 Ca2+依赖性大电导 K+通道。

化合物

Atosiban
Cat.No: T4996
Synonym: 阿托西班,RWJ22164,RW22164
Target: Oxytocin Receptor, Vasopressin Receptor
Atosiban acetate
Cat.No: T5148
Synonym: RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164,醋酸阿托西班
Target: Oxytocin Receptor, Vasopressin Receptor
SSR126768A
Cat.No: T28855
Synonym: SSR-126768A,SSR 126768A
Target: Oxytocin Receptor
Erlosiban
Cat.No: T70570
Synonym:
Target:
Ebopiprant HCl
Cat.No: T70000
Synonym:
Target:
11,12-DiHETrE
Cat.No: T73762
Synonym:
Target:
PDC31
Cat.No: T76565
Synonym:
Target:
TargetMol Loading
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