Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T78714 |
PptT-IN-4
|
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
PptT-IN-4 (Compound 3a) 为PptT抑制剂,IC50为0.71 μM。其对MtbH37Rv的MIC值为42 μM,并且还能抑制hERG、hCav1.2和hNav1.5通道,对应IC50s分别为11 μM、8.1 μM、6.9 μM。 |