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抑制剂 & 化合物

4

天然产物

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Cat. No. Product Name Target Signaling Pathways
T7535 RGX-202

胍基丙酸,β-GPA,3-Guanidinopropionic Acid

AMPK; PPAR Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism; PI3K/Akt/mTOR signaling
RGX-202 (β-GPA) 是口服有活性的SLC6A8转运蛋白抑制剂。它在体内外均能够强烈地抑制肌酸输入,降低细胞内磷酸肌酸和 ATP 水平,诱导肿瘤凋亡,可于研究肿瘤。
T76113 Creatine kinase (OcCK)

Creatine kinase (OcCK) 催化肌酸和 ATP 的可逆反应,形成磷酸肌酸和 ADP。Creatine kinase (OcCK) 是在快速能量周转期间维持恒定 ATP/ADP 比率的关键酶。

化合物

RGX-202
Cat.No: T7535
Synonym: 胍基丙酸,β-GPA,3-Guanidinopropionic Acid
Target: AMPK, PPAR
Creatine kinase (OcCK)
Cat.No: T76113
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T3262 Phosphocreatine disodium

Disodium phosphocreatine,Phosphocreatine disodium salt,Creatine phosphate disodium salt,磷酸肌酸钠

Others; Endogenous Metabolite Metabolism; Others
Phosphocreatine disodium (Phosphocreatine disodium salt) 是一种磷酸化的肌酸分子,在肌肉、骨骼和大脑中作为一种可快速动员的高能磷酸盐储备。
T4888 Phosphocreatine disodium hydrate

磷酸肌酸二钠盐,Phosphocreatine disodium salt hydrate

Others; Endogenous Metabolite Metabolism; Others
Phosphocreatine disodium hydrate 是内源性代谢产物的一种。
T19515 Phosphocreatine dipotassium

Creatinephosphoric acid (dipotassium),Creatine phosphate (dipotassium)

Others Others
Phosphocreatine dipotassium, primarily found in the skeletal muscles of vertebrates and one of organic compounds known as alpha amino acids and derivatives.
T4883 Creatine

Methylguanidoacetic acid,肌酸

Endogenous Metabolite Metabolism
Creatine (Methylguanidoacetic acid) 是一种内源性氨基酸代谢物,在细胞能量中发挥重要作用,尤其是在肌肉和大脑中。

天然产物

Phosphocreatine disodium
Cat.No: T3262
Synonym: Disodium phosphocreatine,Phosphocreatine disodium salt,Creatine phosphate disodium salt,磷酸肌酸钠
Target: Others, Endogenous Metabolite
Phosphocreatine disodium hydrate
Cat.No: T4888
Synonym: 磷酸肌酸二钠盐,Phosphocreatine disodium salt hydrate
Target: Others, Endogenous Metabolite
Phosphocreatine dipotassium
Cat.No: T19515
Synonym: Creatinephosphoric acid (dipotassium),Creatine phosphate (dipotassium)
Target: Others
Creatine
Cat.No: T4883
Synonym: Methylguanidoacetic acid,肌酸
Target: Endogenous Metabolite
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