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Cat. No. Product Name Target Signaling Pathways
T8767 PfDHODH-IN-2

Dehydrogenase; Parasite Metabolism; Microbiology/Virology
PfDHODH-IN-2 是一种二氢噻吩酮衍生物,是一种有效的恶性疟原虫二氢乳清酸脱氢酶抑制剂,其IC50值为 1.11 µM。它具有抗疟作用,可研究疟疾。
T12438 PfDHODH-IN-1

Dehydrogenase; Parasite Metabolism; Microbiology/Virology
PfDHODH-IN-1 是 Leflunomide 活性代谢物的类似物,具有抗疟疾活性。它是恶性疟原虫二氢乳清酸脱氢酶抑制剂。
T11027 DHODH-IN-4

Dehydrogenase Metabolism
DHODH-IN-4 是人和 Plasmodium falciparum 二氢乳清酸脱氢酶 (DHODH) 的抑制剂,其对 PfDHODH 和 HsDHODH 的IC50 值分别为 4 μM 和 0.18 μM。DHODH-IN-4 (compound 17) 具有抗疟疾活性。
T71061 DSM267

DSM267 is a novel Plasmodium falciparum Dihydroorotate Dehydrogenase (PfDHODH) Inhibitor.
T25524 IDI-3783

IDI-3783 is a mutant-selective inhibitor of Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH).
T25448 Genz-669178

Genz-669178 is a wild-type inhibitor of Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH).
T24122 GW648495

DSM-1,GW-648495,DSM 1,GW 648495,DSM1

GW648495 is a PfDHODH inhibitor that shows greater than 4,000-fold selectivity for the malarial enzyme.
T26900 BRD7539

BRD-7539,BRD 7539

BRD7539B is a Dihydroorotate dehydrogenase (DHODH) inhibitor . RD7539 shows to target PfDHODH (IC50 = 0.033 μM) selectively over human (Hs) DHODH (IC50 > 50 μM).
T15173 DSM265

PfSPZ

Dehydrogenase; Parasite Metabolism; Microbiology/Virology
DSM265 (PfSPZ) 是一种具有抗疟活性的二氢乳清酸脱氢酶抑制剂(IC50:8.9 nM)。DSM265 抑制 Pf3D7 寄生虫的生长可用于治疗和预防疟疾感染。

化合物

PfDHODH-IN-2
Cat.No: T8767
Synonym:
Target: Dehydrogenase, Parasite
PfDHODH-IN-1
Cat.No: T12438
Synonym:
Target: Dehydrogenase, Parasite
DHODH-IN-4
Cat.No: T11027
Synonym:
Target: Dehydrogenase
DSM267
Cat.No: T71061
Synonym:
Target:
IDI-3783
Cat.No: T25524
Synonym:
Target:
Genz-669178
Cat.No: T25448
Synonym:
Target:
GW648495
Cat.No: T24122
Synonym: DSM-1,GW-648495,DSM 1,GW 648495,DSM1
Target:
BRD7539
Cat.No: T26900
Synonym: BRD-7539,BRD 7539
Target:
DSM265
Cat.No: T15173
Synonym: PfSPZ
Target: Dehydrogenase, Parasite
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