Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8767 |
PfDHODH-IN-2
|
Dehydrogenase; Parasite | Metabolism; Microbiology/Virology |
PfDHODH-IN-2 是一种二氢噻吩酮衍生物,是一种有效的恶性疟原虫二氢乳清酸脱氢酶抑制剂,其IC50值为 1.11 µM。它具有抗疟作用,可研究疟疾。 | |||
T12438 |
PfDHODH-IN-1
|
Dehydrogenase; Parasite | Metabolism; Microbiology/Virology |
PfDHODH-IN-1 是 Leflunomide 活性代谢物的类似物,具有抗疟疾活性。它是恶性疟原虫二氢乳清酸脱氢酶抑制剂。 | |||
T11027 |
DHODH-IN-4
|
Dehydrogenase | Metabolism |
DHODH-IN-4 是人和 Plasmodium falciparum 二氢乳清酸脱氢酶 (DHODH) 的抑制剂,其对 PfDHODH 和 HsDHODH 的IC50 值分别为 4 μM 和 0.18 μM。DHODH-IN-4 (compound 17) 具有抗疟疾活性。 | |||
T71061 | DSM267 | ||
DSM267 is a novel Plasmodium falciparum Dihydroorotate Dehydrogenase (PfDHODH) Inhibitor. | |||
T25524 | IDI-3783 | ||
IDI-3783 is a mutant-selective inhibitor of Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH). | |||
T25448 | Genz-669178 | ||
Genz-669178 is a wild-type inhibitor of Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH). | |||
T24122 |
GW648495
DSM-1,GW-648495,DSM 1,GW 648495,DSM1 |
||
GW648495 is a PfDHODH inhibitor that shows greater than 4,000-fold selectivity for the malarial enzyme. | |||
T26900 |
BRD7539
BRD-7539,BRD 7539 |
||
BRD7539B is a Dihydroorotate dehydrogenase (DHODH) inhibitor . RD7539 shows to target PfDHODH (IC50 = 0.033 μM) selectively over human (Hs) DHODH (IC50 > 50 μM). | |||
T15173 |
DSM265
PfSPZ |
Dehydrogenase; Parasite | Metabolism; Microbiology/Virology |
DSM265 (PfSPZ) 是一种具有抗疟活性的二氢乳清酸脱氢酶抑制剂(IC50:8.9 nM)。DSM265 抑制 Pf3D7 寄生虫的生长可用于治疗和预防疟疾感染。 |